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Found 13 Enz. Inhib. hit(s) with all data for entry = 6781
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152509((4-Bromo-2,5-dihydroxyphenyl)(4-hydroxyphenyl)meth...)
Affinity DataKi:  2.78nM IC50:  4.58nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152510((4-Bromo-2,5-dihydroxyphenyl)(phenyl)methanone (23...)
Affinity DataKi:  3.24nM IC50:  4.88nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152500((2-bromo-4-methoxyphenyl)(3,4-dimethoxyphenyl)meth...)
Affinity DataKi:  3.53nM IC50:  4.41nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152506((5-bromo-2,4-dimethoxyphenyl)(4-methoxyphenyl)meth...)
Affinity DataKi:  3.65nM IC50:  4.05nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152508((2-Bromo-4-hydroxyphenyl)(2,3-dihydroxyphenyl)meth...)
Affinity DataKi:  3.75nM IC50:  4.84nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152503((4-Bromo-2,5-dimethoxyphenyl)(4-methoxyphenyl)meth...)
Affinity DataKi:  3.77nM IC50:  4.22nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152507((2-bromo-4-hydroxyphenyl)(3,4-dihydroxyphenyl)meth...)
Affinity DataKi:  4.06nM IC50:  4.71nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152502(2-bromo-1,4-dimethoxybenzene (14))
Affinity DataKi:  4.25nM IC50:  7.21nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152501((2-Bromo-4-methoxyphenyl)(2,3-dimethoxyphenyl)meth...)
Affinity DataKi:  4.34nM IC50:  4.20nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152504((4-Bromo-2,5-dimethoxyphenyl)(phenyl)methanone (16...)
Affinity DataKi:  5.28nM IC50:  4.68nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152511((5-Bromo-2,4-dihydroxyphenyl)(4-hydroxyphenyl)meth...)
Affinity DataKi:  5.72nM IC50:  4.81nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM152505((2,4-dimethoxyphenyl)(4-methoxyphenyl)methanone (1...)
Affinity DataKi:  5.88nM IC50:  5.25nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Ataturk University

LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataKi:  7.64nM IC50:  7.53nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 無 of Tris/HCl buffer (...More data for this Ligand-Target Pair