Compile Data Set for Download or QSAR
maximum 50k data
Found 61 Enz. Inhib. hit(s) with all data for entry = 50046460
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113872(CHEMBL3605139)
Affinity DataIC50:  200nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113937(CHEMBL3605119)
Affinity DataIC50:  400nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113830(CHEMBL3605140)
Affinity DataIC50:  400nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113943(CHEMBL3605004)
Affinity DataIC50:  500nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113833(CHEMBL3605145)
Affinity DataIC50:  500nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113941(CHEMBL3605002)
Affinity DataIC50:  600nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113844(CHEMBL3605123)
Affinity DataIC50:  700nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113836(CHEMBL3605147)
Affinity DataIC50:  700nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113949(CHEMBL3605012)
Affinity DataIC50:  900nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113935(CHEMBL3605117)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113834(CHEMBL3605146)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113945(CHEMBL3605006)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113848(CHEMBL3605127)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113842(CHEMBL3605122)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113841(CHEMBL3605121)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113846(CHEMBL3605126)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113853(CHEMBL3605130)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113876(CHEMBL3605015)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113838(CHEMBL3605120)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch express method based electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113852(CHEMBL3605129)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113890(CHEMBL3605021)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113887(CHEMBL3605019)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113832(CHEMBL3605143)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113875(CHEMBL3605014)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113871(CHEMBL3605138)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113948(CHEMBL3605011)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113922(CHEMBL3605025)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113858(CHEMBL3605132)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113845(CHEMBL3605125)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113870(CHEMBL3605137)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113862(CHEMBL3605134)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113866(CHEMBL3605135)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113930(CHEMBL3605026)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113915(CHEMBL3605024)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113947(CHEMBL3605010)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113850(CHEMBL3605128)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113881(CHEMBL3605016)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113856(CHEMBL3605131)
Affinity DataIC50:  1.22E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113837(CHEMBL3605148)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113861(CHEMBL3605133)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113885(CHEMBL3605017)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50068000(CHEMBL3305167)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch express method based electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113888(CHEMBL3605020)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113886(CHEMBL3605018)
Affinity DataIC50:  2.44E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113838(CHEMBL3605120)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113939(CHEMBL3605000)
Affinity DataIC50:  2.54E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50068000(CHEMBL3305167)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113905(CHEMBL3605022)
Affinity DataIC50:  2.91E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113950(CHEMBL3605013)
Affinity DataIC50:  2.97E+4nMAssay Description:Inhibition of human ERG assessed as reduction in MK499 competitive bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50113950(CHEMBL3605013)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch express method based electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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