Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 50046646
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123357(CHEMBL3622695)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123400(CHEMBL3623256)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123404(CHEMBL3623250)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of human SIRT2 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123400(CHEMBL3623256)
Affinity DataIC50:  1.02E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017341(CHEMBL3288034)
Affinity DataIC50:  1.06E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017341(CHEMBL3288034)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of human SIRT2 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123451(CHEMBL3623255)
Affinity DataIC50:  1.27E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017341(CHEMBL3288034)
Affinity DataIC50:  1.36E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123372(CHEMBL3623251)
Affinity DataIC50:  1.37E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123372(CHEMBL3623251)
Affinity DataIC50:  1.37E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123357(CHEMBL3622695)
Affinity DataIC50:  1.59E+5nMAssay Description:Inhibition of human SIRT2 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123357(CHEMBL3622695)
Affinity DataIC50:  2.38E+5nMAssay Description:Inhibition of human SIRT1 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123403(CHEMBL3623259)
Affinity DataIC50:  2.42E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  2.42E+5nMAssay Description:Inhibition of human SIRT2 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123401(CHEMBL3623257)
Affinity DataIC50:  2.70E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123401(CHEMBL3623257)
Affinity DataIC50:  2.75E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123403(CHEMBL3623259)
Affinity DataIC50:  2.97E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123452(CHEMBL3623260)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50017341(CHEMBL3288034)
Affinity DataIC50:  3.14E+5nMAssay Description:Inhibition of human SIRT1 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123364(CHEMBL3622696)
Affinity DataIC50:  4.24E+5nMAssay Description:Inhibition of human SIRT1 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123402(CHEMBL3623258)
Affinity DataIC50:  4.41E+5nMAssay Description:Inhibition of human SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123448(CHEMBL3623253)
Affinity DataIC50:  5.17E+5nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123405(CHEMBL3623252)
Affinity DataIC50:  2.87E+6nMAssay Description:Inhibition of human recombinant SIRT6 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL
LigandPNGBDBM50123399(CHEMBL3623254)
Affinity DataIC50:  6.52E+6nMAssay Description:Inhibition of human SIRT1 deacetylase activity using Arg-His-Lys-Lys(AC)-AMC as a substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed