Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50046618
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50121656(CHEMBL3616869)
Affinity DataIC50:  5.21E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human CDK2 (1 to 298 amino acid residues) expressed in Escherichia coli BL21 assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50121656(CHEMBL3616869)
Affinity DataIC50:  5.51E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human CDK2 (1 to 298 amino acid residues) expressed in Escherichia coli BL21 assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50121656(CHEMBL3616869)
Affinity DataIC50:  5.82E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human CDK2 (1 to 298 amino acid residues) expressed in Escherichia coli BL21 assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50121656(CHEMBL3616869)
Affinity DataIC50:  6.98E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human CDK2 (1 to 298 amino acid residues) expressed in Escherichia coli BL21 assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50121656(CHEMBL3616869)
Affinity DataIC50:  7.83E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human CDK2 (1 to 298 amino acid residues) expressed in Escherichia coli BL21 assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50121658(CHEMBL3616877)
Affinity DataIC50:  1.05E+5nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human CDK2 (1 to 298 amino acid residues) expressed in Escherichia coli BL21 assessed as inhibi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50121656(CHEMBL3616869)
Affinity DataIC50:  1.51E+5nMAssay Description:Binding affinity to human CDK2 Y180A mutant expressed in Escherichia coli BL21 assessed as inhibition of interaction with cyclin A3 by measuring HHAS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50121656(CHEMBL3616869)
Affinity DataIC50:  8.85E+5nMAssay Description:Binding affinity to human CDK2 R150A mutant expressed in Escherichia coli BL21 assessed as inhibition of interaction with cyclin A3 by measuring HHAS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed