Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 7215
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
The University Of Kansas Medical Center

LigandPNGBDBM181109(3-Mercaptopicolinic acid (MPA))
Affinity DataKi:  3.70E+4nM ΔG°:  -25.3kJ/moleT: 2°CAssay Description:OAA/PEP binding site. When the enzyme was assayed in the direction of PEP →OAA, the standard reaction mixture contained 50 mM HEPES (pH 7.5), 2...More data for this Ligand-Target Pair
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
The University Of Kansas Medical Center

LigandPNGBDBM181109(3-Mercaptopicolinic acid (MPA))
Affinity DataKi:  4.50E+4nM ΔG°:  -24.8kJ/moleT: 2°CAssay Description:OAA/PEP binding site. The activity of PEPCK in the direction from OAA to PEP was assayed with 50 mM HEPES (pH 7.5), 10 mM DTT, 4 mM MgCl2, 0.5 mM GTP...More data for this Ligand-Target Pair
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
The University Of Kansas Medical Center

LigandPNGBDBM181109(3-Mercaptopicolinic acid (MPA))
Affinity DataKi:  8.30E+4nM ΔG°:  -23.3kJ/moleT: 2°CAssay Description:Allosteric binding site. When the enzyme was assayed in the direction of PEP →OAA, the standard reaction mixture contained 50 mM HEPES (pH 7.5)...More data for this Ligand-Target Pair
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
The University Of Kansas Medical Center

LigandPNGBDBM181109(3-Mercaptopicolinic acid (MPA))
Affinity DataKi:  8.30E+4nM ΔG°:  -23.3kJ/moleT: 2°CAssay Description:OAA/PEP binding site. When the enzyme was assayed in the direction of PEP →OAA, the standard reaction mixture contained 50 mM HEPES (pH 7.5), 2...More data for this Ligand-Target Pair
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
The University Of Kansas Medical Center

LigandPNGBDBM181109(3-Mercaptopicolinic acid (MPA))
Affinity DataKi:  1.21E+5nM ΔG°:  -22.4kJ/moleT: 2°CAssay Description:Allosteric binding site. The activity of PEPCK in the direction from OAA to PEP was assayed with 50 mM HEPES (pH 7.5), 10 mM DTT, 4 mM MgCl2, 0.5 mM ...More data for this Ligand-Target Pair
TargetPhosphoenolpyruvate carboxykinase, cytosolic [GTP](Rattus norvegicus (Rat))
The University Of Kansas Medical Center

LigandPNGBDBM181109(3-Mercaptopicolinic acid (MPA))
Affinity DataKi:  1.80E+5nM ΔG°:  -21.4kJ/moleT: 2°CAssay Description:Allosteric binding site. When the enzyme was assayed in the direction of PEP →OAA, the standard reaction mixture contained 50 mM HEPES (pH 7.5)...More data for this Ligand-Target Pair