Found 34 Enz. Inhib. hit(s) with all data for entry = 50046676 
Affinity DataKi: 0.0300nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of KLK7 (unknown origin) expressed in Pichia pastoris X33 using KHLY-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of KLK4 (unknown origin) expressed in Sf9 cells using FVQRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of KLK7 (unknown origin) expressed in Pichia pastoris X33 using KHLY-pNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of KLK4 (unknown origin) expressed in Sf9 cells using FVQRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetTransmembrane protease serine 6(Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Inhibition of matriptase (unknown origin) using Ac-RQFRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetTransmembrane protease serine 6(Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 87nMAssay Description:Inhibition of matriptase (unknown origin) using Ac-RQFRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 214nMAssay Description:Inhibition of alpha-thrombin (unknown origin) using Ac-ATPRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 362nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 379nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Inhibition of alpha-thrombin (unknown origin) using Ac-ATPRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetTransmembrane protease serine 6(Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 546nMAssay Description:Inhibition of matriptase (unknown origin) using Ac-RQFRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 549nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.83E+3nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetTransmembrane protease serine 6(Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.36E+4nMAssay Description:Inhibition of matriptase (unknown origin) using Ac-RQFRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.43E+4nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.71E+4nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetTransmembrane protease serine 6(Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.93E+4nMAssay Description:Inhibition of matriptase (unknown origin) using Ac-RQFRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of alpha-thrombin (unknown origin) using Ac-ATPRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of alpha-thrombin (unknown origin) using Ac-ATPRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
TargetTransmembrane protease serine 6(Homo sapiens (Human))
Queensland University Of Technology
Curated by ChEMBL
Queensland University Of Technology
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of matriptase (unknown origin) using Ac-RQFRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
