Found 15 Enz. Inhib. hit(s) with all data for entry = 50046597 TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 5.30E+3nMAssay Description:Allosteric modulation of GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 3.32E+4nMAssay Description:Partial agonist activity at GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as induction of chloride c...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 2.15E+4nMAssay Description:Allosteric modulation of GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 1.58E+4nMAssay Description:Allosteric modulation of GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 2.46E+4nMAssay Description:Allosteric modulation of GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Allosteric modulation of GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 2.04E+4nMAssay Description:Allosteric modulation of GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 1.44E+4nMAssay Description:Allosteric modulation of GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 5.10E+4nMAssay Description:Partial agonist activity at GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as induction of chloride c...More data for this Ligand-Target Pair
3D Structure (crystal)TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 7.62E+4nMAssay Description:Partial agonist activity at GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as induction of chloride c...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 6.81E+4nMAssay Description:Partial agonist activity at GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as induction of chloride c...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 1.44E+5nMAssay Description:Partial agonist activity at GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as induction of chloride c...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 6.22E+4nMAssay Description:Partial agonist activity at GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as induction of chloride c...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 6.90E+3nMAssay Description:Partial agonist activity at GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as induction of chloride c...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Graz
Curated by ChEMBL
University Of Graz
Curated by ChEMBL
Affinity DataEC50: 4.76E+4nMAssay Description:Allosteric modulation of GABAAalpha1beta2gamma2s receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induc...More data for this Ligand-Target Pair
