Compile Data Set for Download or QSAR
maximum 50k data
Found 37 Enz. Inhib. hit(s) with all data for entry = 50046922
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138221(CHEMBL3752627)
Affinity DataIC50:  9nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138221(CHEMBL3752627)
Affinity DataIC50:  9nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138221(CHEMBL3752627)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced inhibition of calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138221(CHEMBL3752627)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced inhibition of chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138224(CHEMBL3753813)
Affinity DataIC50:  36nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138224(CHEMBL3753813)
Affinity DataIC50:  36nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138242(CHEMBL3751958)
Affinity DataIC50:  69nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138243(CHEMBL3753826)
Affinity DataIC50:  114nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138227(CHEMBL3752690)
Affinity DataIC50:  150nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138226(CHEMBL3753161)
Affinity DataIC50:  210nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138241(CHEMBL3754764)
Affinity DataIC50:  249nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138253(CHEMBL3754334)
Affinity DataIC50:  254nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138254(CHEMBL3752224)
Affinity DataIC50:  284nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138247(CHEMBL3753178)
Affinity DataIC50:  301nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138248(CHEMBL3752640)
Affinity DataIC50:  328nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138258(CHEMBL3754037)
Affinity DataIC50:  438nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138249(CHEMBL3754155)
Affinity DataIC50:  550nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138277(CHEMBL3754119)
Affinity DataIC50:  700nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138246(CHEMBL3751959)
Affinity DataIC50:  744nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138255(CHEMBL3753719)
Affinity DataIC50:  928nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138260(CHEMBL3753478)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138252(CHEMBL3753563)
Affinity DataIC50:  1.69E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138251(CHEMBL3754349)
Affinity DataIC50:  2.64E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138275(CHEMBL3753509)
Affinity DataIC50:  2.97E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138276(CHEMBL3754549)
Affinity DataIC50:  3.42E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138245(CHEMBL3751926)
Affinity DataIC50:  3.48E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138250(CHEMBL3752652)
Affinity DataIC50:  3.70E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138256(CHEMBL3753474)
Affinity DataIC50:  3.70E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138222(CHEMBL3753491)
Affinity DataIC50:  4.50E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138229(CHEMBL3752915)
Affinity DataIC50:  5.41E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138223(CHEMBL3753526)
Affinity DataIC50:  5.78E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138225(CHEMBL3753005)
Affinity DataIC50:  6.15E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138228(CHEMBL3753428)
Affinity DataIC50:  6.61E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138259(CHEMBL3753683)
Affinity DataIC50:  8.20E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138257(CHEMBL3752110)
Affinity DataIC50:  9.74E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138274(CHEMBL3752614)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138244(CHEMBL3752398)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed