Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50047015
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143549(CHEMBL3758801)
Affinity DataIC50:  130nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143555(CHEMBL3759729)
Affinity DataIC50:  650nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143554(CHEMBL3758708)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143550(CHEMBL3759902)
Affinity DataIC50:  2.56E+3nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143548(CHEMBL3759783)
Affinity DataIC50:  5.98E+3nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143547(CHEMBL3759248)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143545(CHEMBL3759818)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143552(CHEMBL3759664)
Affinity DataIC50:  2.95E+4nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143600(CHEBI:29571 | Dehydroabietic Acid)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143553(CHEMBL3759966)
Affinity DataIC50:  4.09E+4nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143551(CHEMBL3759598)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143546(CHEMBL3760052)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed