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Found 94 Enz. Inhib. hit(s) with all data for entry = 50047459
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168215(CHEMBL3804916)
Affinity DataKi:  250nMAssay Description:Reversible inhibition of human estrone sulfatase using 4-methylumbelliferyl sulfate as substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50112876(3-((N-cyclohexyl-aminocarbonoyl)hydrazono]methyl)-...)
Affinity DataKi:  350nMAssay Description:Non-competitive inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 20 mins by Lineweaver-Burk plot a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50151137(2-Adamantan-1-yl-4-oxo-4H-thiochromene-6-carboxyli...)
Affinity DataKi:  500nMAssay Description:Reversible inhibition of recombinant human estrone sulfatase using 4-methylumbelliferyl sulfate as substrate by Hanes plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168258(CHEMBL3805369)
Affinity DataKi:  890nMAssay Description:Inhibition of recombinant human estrone sulfatase expressed in CHO cells using 4-methylumbelliferyl sulfate as substrate by Hanes plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168216(CHEMBL3806006)
Affinity DataKi:  2.80E+3nMAssay Description:Reversible inhibition of human estrone sulfatase using 4-methylumbelliferyl sulfate as substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168214(CHEMBL3806064)
Affinity DataKi:  8.20E+4nMAssay Description:Reversible inhibition of estrone sulfatase (unknown origin) using 4-methylumbelliferyl sulfate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168219(CHEMBL3805209)
Affinity DataIC50:  0.0240nMAssay Description:Inhibition of estrone sulfatase (unknown origin) transfected in HEK293 cells using E1S as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168217(CHEMBL3806018)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of estrone sulfatase (unknown origin) transfected in HEK293 cells using E1S as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50380223(CHEMBL2011422)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of placental microsomal estrone sulfatase (unknown origin) using [6,7-3H]E1S as substrate incubated for 1 hr by scintillation spectrometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50369432(CHEMBL1627465)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of human placental estrone sulfatase expressed in HEK293 cells using [3H]E1S as substrate incubated for 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50136297(CHEMBL136112 | Sulfamic acid 2-adamantan-2-ylidene...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of estrone sulfatase in human sebocytes using DHEAS as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50118560(CHEMBL262050 | Sulfamic acid 2-adamantan-1-yl-4-ox...)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of recombinant human estrone sulfatase using 4-methylumbelliferyl sulfate as substrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168259(CHEMBL3806300)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human placental estrone sulfatase expressed in HEK293 cells using [3H]E1S as substrate incubated for 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50136297(CHEMBL136112 | Sulfamic acid 2-adamantan-2-ylidene...)
Affinity DataIC50:  0.75nMAssay Description:Inhibition of estrone sulfatase human keratinocytes using DHEAS as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50136297(CHEMBL136112 | Sulfamic acid 2-adamantan-2-ylidene...)
Affinity DataIC50:  0.770nMAssay Description:Inhibition of estrone sulfatase in human MCF7 cells using estrone sulphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human placental estrone sulfatase expressed in HEK293 cells using [3H]E1S as substrate incubated for 2 hrs by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121065(CHEMBL3622012)
Affinity DataIC50:  1nMAssay Description:Inhibition of placental microsomal estrone sulfatase (unknown origin) using [3H]-estrone sulphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121113(CHEMBL3622018)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121116(CHEMBL3622021)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121117(CHEMBL3622022)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121192(CHEMBL1235380)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121195(CHEMBL3622028)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121193(CHEMBL3622026)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121194(CHEMBL3622027)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121174(CHEMBL3622024)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121119(CHEMBL3622023)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121118(CHEMBL3621214)
Affinity DataIC50:  1nMAssay Description:Inhibition of human placental microsomal estrone sulfatase using [3H]E1S as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50369431(CHEMBL1627878)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of estrone sulfatase (unknown origin) transfected in HEK293 cells using [3H]E1S as substrate incubated for 2 hrs by liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of estrone sulfatase (unknown origin) transfected in HEK293 cells using [3H]E1S as substrate incubated for 2 hrs by liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50136297(CHEMBL136112 | Sulfamic acid 2-adamantan-2-ylidene...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of estrone sulfatase in human skin fibroblasts using DHEAS as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 4 hrs by liquid scintillation counting me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM13058(6-oxo-6,7,8,9,10,11-hexahydrocyclohepta[c]chromen-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of placental microsomal estrone sulfatase (unknown origin) using [3H]-estrone sulphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168220(CHEMBL3805984)
Affinity DataIC50:  9nMAssay Description:Inhibition of estrone sulfatase in human MCF7 cells using [3H]E1S as substrate incubated for 24 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of placental microsomal estrone sulfatase (unknown origin) using [6,7-3H]E1S as substrate incubated for 1 hr by scintillation spectrometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50121059(CHEMBL3622030)
Affinity DataIC50:  10nMAssay Description:Inhibition of estrone sulfatase in human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50366532(CHEMBL518966)
Affinity DataIC50:  12nMAssay Description:Inhibition of estrone sulfatase (unknown origin) transfected in HEK293 cells using [3H]E1S as substrate incubated for 2 hrs by liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168224(CHEMBL3805967)
Affinity DataIC50:  14nMAssay Description:Inhibition of estrone sulfatase (unknown origin) transfected in HEK293 cells using [3H]E1S as substrate incubated for 2 hrs by liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168221(CHEMBL3805064)
Affinity DataIC50:  21nMAssay Description:Inhibition of estrone sulfatase (unknown origin) transfected in HEK293 cells using [3H]E1S as substrate incubated for 2 hrs by liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  25nMAssay Description:Inhibition of placental microsomal estrone sulfatase (unknown origin) using [3H]-estrone sulphate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168231(CHEMBL3806175)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168230(CHEMBL3805387)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168229(CHEMBL3806088)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168233(CHEMBL3805071)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168245(CHEMBL3806272)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168251(CHEMBL3805959)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168252(CHEMBL3805117)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168253(CHEMBL3806025)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168254(CHEMBL3805811)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50168256(CHEMBL3805090)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50369432(CHEMBL1627465)
Affinity DataIC50:  30nMAssay Description:Inhibition of estrone sulfatase in human JEG-3 cells using [3H]-estrone sulphate as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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