Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [3H]W-7 from bovine brain CaMMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Binding affinity to CaM (unknown origin) by equilibrium dialysis methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Displacement of [3H]trifluoperazine from bovine brain CaM in presence of calciumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+4nMAssay Description:Displacement of [3H] ifenprodil from bovine CaM-agarose incubated for 30 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Binding affinity to CaM (unknown origin) by equilibrium dialysis methodMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 4.04E+4nMAssay Description:Inhibition of full length recombinant human CaMKK2 expressed in insect Sf21 cells in presence of 2 uM CaM/[gamma32P]ATP by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+4nMAssay Description:Binding affinity to CaM (unknown origin) by equilibrium dialysis methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+5nMAssay Description:Competitive binding affinity to human recombinant CaM by Cy5 dye labeled W-7-based fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataKd: 470nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Binding affinity to dansylated bovine testes CaM by fluorescence analysis in presence of calcium2+More data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Binding affinity to dansylated bovine testes CaM by fluorescence analysis in presence of calcium2+More data for this Ligand-Target Pair
Affinity DataKd: 7.20E+3nMAssay Description:Binding affinity to dansylated bovine testes CaM by fluorescence analysis in presence of calcium2+More data for this Ligand-Target Pair
Affinity DataKd: 850nMAssay Description:Binding affinity to CaM (unknown origin) by isothermal titration calorimetric analysis in presence of calcium2+More data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Binding affinity to dansylated bovine brain CaM assessed as half maximal increase in fluorescence by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 7.20E+3nMAssay Description:Binding affinity to dansylated bovine brain CaM assessed as half maximal increase in fluorescence by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataKd: 5.00E+3nMAssay Description:Binding affinity to dansylated bovine testes CaM by fluorescence analysis in presence of calcium2+More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMAssay Description:Binding affinity to dansylated bovine brain CaM assessed as half maximal increase in fluorescence by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataKd: 2.90E+3nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 6.10E+4nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+4nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 5.00E+4nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 3.10E+3nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 3.50E+3nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 2.90E+3nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 3.40E+3nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to bovine brain CaM by FTPFACE analysisMore data for this Ligand-Target Pair