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Found 52 Enz. Inhib. hit(s) with all data for entry = 50047495
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM32142(5-amino-8-quinolinol | 5-aminoquinolin-8-ol | 5-az...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human MDAY-D2 cells assessed as free 7-ami...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM32142(5-amino-8-quinolinol | 5-aminoquinolin-8-ol | 5-az...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human K562 cells assessed as free 7-amino-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM32142(5-amino-8-quinolinol | 5-aminoquinolin-8-ol | 5-az...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human KG1A cells assessed as free 7-amino-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM32142(5-amino-8-quinolinol | 5-aminoquinolin-8-ol | 5-az...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human NB4 cells assessed as free 7-amino-4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM32142(5-amino-8-quinolinol | 5-aminoquinolin-8-ol | 5-az...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human OCI-AML2 cells assessed as free 7-am...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM32142(5-amino-8-quinolinol | 5-aminoquinolin-8-ol | 5-az...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human KMS18 cells assessed as free 7-amino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM32142(5-amino-8-quinolinol | 5-aminoquinolin-8-ol | 5-az...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human KMH11 cells assessed as free 7-amino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM32142(5-amino-8-quinolinol | 5-aminoquinolin-8-ol | 5-az...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate expressed in human UTMC2 cells assessed as free 7-amino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171081(CHEMBL3805036)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate assessed as fluorescence quinching control by fluoresce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50170997(CHEMBL3805801)
Affinity DataIC50:  5.26E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171045(CHEMBL3805324)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50170999(CHEMBL3805496)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171000(CHEMBL3805486)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171001(CHEMBL3805988)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171046(CHEMBL3805440)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171002(CHEMBL3806320)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171047(CHEMBL3805100)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171034(CHEMBL3805013)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171003(CHEMBL3805932)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50170998(CHEMBL3805812)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171006(CHEMBL3805160)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171080(CHEMBL3806316)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50170997(CHEMBL3805801)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of human 20S proteasome caspase beta1-like activity using Z-LLE-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171036(CHEMBL3805729)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171038(CHEMBL3805213)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171039(CHEMBL3806263)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171044(CHEMBL3805167)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171038(CHEMBL3805213)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibition of human 20S proteasome caspase beta1-like activity using Z-LLE-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171079(CHEMBL3805403)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171040(CHEMBL3805282)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171037(CHEMBL3806156)
Affinity DataIC50:  1.99E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171082(CHEMBL3805379)
Affinity DataIC50:  2.16E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171041(CHEMBL3805307)
Affinity DataIC50:  2.36E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171033(CHEMBL3806104)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171005(CHEMBL3804889)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171004(CHEMBL3805918)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171032(CHEMBL3805787)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171031(CHEMBL3804977)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171008(CHEMBL3805485)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50170997(CHEMBL3805801)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome tryptic beta2-like activity using Z-ARR-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171038(CHEMBL3805213)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome tryptic beta2-like activity using Z-ARR-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171084(CHEMBL3805961)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171083(CHEMBL3805152)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171081(CHEMBL3805036)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171078(CHEMBL3804847)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171077(CHEMBL3805957)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171035(CHEMBL3805830)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171043(CHEMBL3805312)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171042(CHEMBL3805672)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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