Affinity DataIC50: 50nMAssay Description:Inhibition of FLAG-tagged mouse JAK1 expressed in insect Sf9 cells using biotin-EQEDEPEGDYFEWLE-NH2 as substrate by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of JAK1 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of JAK1 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of JAK1 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of FLAG-tagged human JAK3 expressed in insect Sf9 cells using biotin-EQEDEPEGDYFEWLE-NH2 as substrate by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of JAK3 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of JAK3 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of JAK3 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of JAK1 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of JAK2 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of JAK2 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of FLAG-tagged human JAK2 expressed in insect Sf9 cells using biotin-EQEDEPEGDYFEWLE-NH2 as substrate by HTRF assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of FLAG-tagged human TYK2 expressed in insect Sf9 cells using biotin-EQEDEPEGDYFEWLE-NH2 as substrate by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of JAK2 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of TYK2 (unknown origin) using tyrosine 3 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of TYK2 (unknown origin) using tyrosine 3 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of JAK1 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of JAK1 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of TYK2 (unknown origin) using tyrosine 3 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of JAK1 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of JAK3 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of JAK2 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of JAK3 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of JAK3 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of JAK2 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.06E+4nMAssay Description:Inhibition of JAK3 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of TYK2 (unknown origin) using tyrosine 3 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.73E+4nMAssay Description:Inhibition of JAK2 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of JAK2 (unknown origin) using tyrosine 6 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataIC50: 3.07E+4nMAssay Description:Inhibition of TYK2 (unknown origin) using tyrosine 3 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of TYK2 (unknown origin) using tyrosine 3 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Konkuk University
Curated by ChEMBL
Konkuk University
Curated by ChEMBL
Affinity DataIC50: 4.22E+4nMAssay Description:Inhibition of TYK2 (unknown origin) using tyrosine 3 peptide as substrate by z'-lyte assayMore data for this Ligand-Target Pair