Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50001838
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018316(2-Butyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018341(2-Ethyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018315(2-Ethynyl-3',4'-dimethoxy-biphenyl-4-carboxylic ac...)
Affinity DataIC50:  5nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018325(CHEMBL53584 | [1,1';2',1'']Terphenyl-4'-carboxylic...)
Affinity DataIC50:  5nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018321(3',4'-Dimethoxy-biphenyl-4-carboxylic acid (1-meth...)
Affinity DataIC50:  15nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018338(2-Butyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  18nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018337(3'-Methoxy-biphenyl-4-carboxylic acid (1-methyl-4-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018320(3',4'-Dimethoxy-2-propyl-biphenyl-4-carboxylic aci...)
Affinity DataIC50:  50nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018324(CHEMBL299760 | [1,1';2',1'']Terphenyl-4'-carboxyli...)
Affinity DataIC50:  50nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018329(3',4'-Dimethoxy-biphenyl-4-carbothioic acid (1-met...)
Affinity DataIC50:  60nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018326(2-Allyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  80nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018322(4,4''-Dimethoxy-[1,1';2',1'']terphenyl-4'-carboxyl...)
Affinity DataIC50:  125nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018336(3',4'-Dimethoxy-biphenyl-4-carbothioic acid (4-pyr...)
Affinity DataIC50:  140nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018327(2-Bromo-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  180nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018323(3,3''-Dimethoxy-[1,1';2',1'']terphenyl-4'-carboxyl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018319(3',4'-Dimethoxy-2-nitro-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  200nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018328(3',4'-Dimethyl-biphenyl-4-carboxylic acid (4-pyrid...)
Affinity DataIC50:  200nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018331(3',4'-Dimethoxy-2-nitro-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  200nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018330(2-Bromo-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  220nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018318(3'-Methoxy-biphenyl-4-carboxylic acid (4-pyridin-3...)
Affinity DataIC50:  280nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018333(2,3',4'-Trimethoxy-biphenyl-4-carboxylic acid (4-p...)
Affinity DataIC50:  300nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018317(3'-Hydroxy-biphenyl-4-carboxylic acid (4-pyridin-3...)
Affinity DataIC50:  300nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018332(3',4'-Dimethoxy-biphenyl-4-carboxylic acid (4-pyri...)
Affinity DataIC50:  400nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018334(3'-Methyl-biphenyl-4-carboxylic acid (4-pyridin-3-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018335(Biphenyl-4-carboxylic acid (4-pyridin-3-yl-butyl)-...)
Affinity DataIC50:  630nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018339(3'-(Cyclohepta-1,3,5-trienyloxy)-biphenyl-4-carbox...)
Affinity DataIC50:  700nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018340(2,3'-Difluoro-biphenyl-4-carboxylic acid (4-pyridi...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed