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Found 18 Enz. Inhib. hit(s) with all data for entry = 50048079
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204010(CHEMBL3928769)
Affinity DataEC50: <300nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells coexpressing NFAT BLA assessed as increase in intracellular Ca2+ flux by fluo-4-AM dye based F...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204016(CHEMBL3959220)
Affinity DataEC50: <10nMAssay Description:Agonist activity at human GPR40 expressed in CHOK cells assessed as increase in intracellular Ca2+ flux by Fluo-4 based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50362690(AMG-837 | CHEMBL1829173)
Affinity DataEC50:  13nMAssay Description:Agonist activity at GPR40 (unknown origin) by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204012(CHEMBL3955132)
Affinity DataEC50:  152nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by calcium-4 dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204013(CHEMBL3900797)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells coexpressing NFAT BLA assessed as increase in intracellular Ca2+ flux by fluo-4-AM dye based F...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204014(CHEMBL3944424 | US10059667, Example 27)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells coexpressing NFAT BLA assessed as increase in intracellular Ca2+ flux by fluo-4-AM dye based F...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50102727(CHEMBL3330550)
Affinity DataEC50:  6nMAssay Description:Agonist activity at GPR40 (unknown origin) by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204015(CHEMBL3954235)
Affinity DataEC50:  10nMAssay Description:Agonist activity at GPR40 (unknown origin) by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204020(CHEMBL3927519)
Affinity DataEC50:  119nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by calcium-4 dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204021(CHEMBL3931755)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells coexpressing NFAT BLA assessed as increase in intracellular Ca2+ flux by fluo-4-AM dye based F...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50200369(CHEMBL3915620)
Affinity DataEC50:  233nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by calcium-4 dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204023(CHEMBL3905856)
Affinity DataEC50:  42nMAssay Description:Agonist activity at flag-tagged human GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204018(CHEMBL3923877)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at rat GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204017(CHEMBL3966288)
Affinity DataEC50: <100nMAssay Description:Agonist activity at full length recombinant human GPR40 expressed in CHOK1 cells assessed as intracellular IP3 accumulation by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204022(CHEMBL3954105)
Affinity DataEC50:  630nMAssay Description:Agonist activity at rat GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204019(CHEMBL3927863)
Affinity DataEC50:  10nMAssay Description:Agonist activity at rat GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204024(CHEMBL3973075)
Affinity DataEC50:  71nMAssay Description:Agonist activity at flag-tagged human GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50204011(CHEMBL3958983)
Affinity DataEC50:  146nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by calcium-4 dye based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed