Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50048192
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207528(CHEMBL3925060)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207530(CHEMBL3930236)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207530(CHEMBL3930236)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207528(CHEMBL3925060)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207531(CHEMBL3897010)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207532(CHEMBL3939235)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207533(CHEMBL3956669)
Affinity DataEC50:  6.17E+4nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207531(CHEMBL3897010)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207534(CHEMBL3957870)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207535(CHEMBL3902257)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207533(CHEMBL3956669)
Affinity DataEC50:  6.10E+4nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207536(CHEMBL3929127)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207537(CHEMBL3911275)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207536(CHEMBL3929127)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207534(CHEMBL3957870)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207538(CHEMBL3931202)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207535(CHEMBL3902257)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207529(CHEMBL3933958)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207532(CHEMBL3939235)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207537(CHEMBL3911275)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207538(CHEMBL3931202)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207529(CHEMBL3933958)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed