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Found 30 Enz. Inhib. hit(s) with all data for entry = 50049033
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429057(CHEMBL2334891)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]SCH23390 from human 3HA-tagged dopamine D1 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429045(CHEMBL1457510)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429057(CHEMBL2334891)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429045(CHEMBL1457510)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429057(CHEMBL2334891)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]SCH23390 from human FLAG-tagged dopamine D3 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429057(CHEMBL2334891)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]SCH23390 from human FLAG-tagged dopamine D2 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429051(CHEMBL2334885)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429045(CHEMBL1457510)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429047((-)-Tetrahydroberberine | CANADINE)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429047((-)-Tetrahydroberberine | CANADINE)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429057(CHEMBL2334891)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D4 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429047((-)-Tetrahydroberberine | CANADINE)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429045(CHEMBL1457510)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424075((-)-Corydalmine | CHEMBL448891)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424077((-)-Tetrahydropalmatine | L-Tetrahydropalmatine | ...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]SCH23390 from human 3HA-tagged dopamine D1 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429051(CHEMBL2334885)
Affinity DataKi:  199nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424075((-)-Corydalmine | CHEMBL448891)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429051(CHEMBL2334885)
Affinity DataKi:  262nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424077((-)-Tetrahydropalmatine | L-Tetrahydropalmatine | ...)
Affinity DataKi:  305nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429051(CHEMBL2334885)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429047((-)-Tetrahydroberberine | CANADINE)
Affinity DataKi:  433nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429047((-)-Tetrahydroberberine | CANADINE)
Affinity DataKi:  486nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424075((-)-Corydalmine | CHEMBL448891)
Affinity DataKi:  533nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424077((-)-Tetrahydropalmatine | L-Tetrahydropalmatine | ...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D4 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429051(CHEMBL2334885)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424075((-)-Corydalmine | CHEMBL448891)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424077((-)-Tetrahydropalmatine | L-Tetrahydropalmatine | ...)
Affinity DataKi:  1.13E+3nMAssay Description:Displacement of [3H]SCH23390 from human FLAG-tagged dopamine D2 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424077((-)-Tetrahydropalmatine | L-Tetrahydropalmatine | ...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [3H]SCH23390 from human FLAG-tagged dopamine D3 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50424075((-)-Corydalmine | CHEMBL448891)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50429045(CHEMBL1457510)
Affinity DataKi:  1.98E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed