Compile Data Set for Download or QSAR
maximum 50k data
Found 55 Enz. Inhib. hit(s) with all data for entry = 50035627
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019624(1-(2-Ethoxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-yl)...)
Affinity DataIC50:  6.10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019595(2-(4-Methyl-piperazin-1-yl)-1-(2-phenoxy-ethyl)-1H...)
Affinity DataIC50:  6.90nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019605(1-(2-Ethoxy-ethyl)-2-(4-pentyl-[1,4]diazepan-1-yl)...)
Affinity DataIC50:  7.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019643(2-(4-Butyl-[1,4]diazepan-1-yl)-1-(2-ethoxy-ethyl)-...)
Affinity DataIC50:  8.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019644(1-(2-Ethoxy-ethyl)-2-(4-propyl-[1,4]diazepan-1-yl)...)
Affinity DataIC50:  8.40nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019602(1-(2-Ethoxy-ethyl)-2-(4-hexyl-piperazin-1-yl)-1H-b...)
Affinity DataIC50:  8.60nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019628(2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-phenoxy-ethyl...)
Affinity DataIC50:  9.10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019609(2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-prop-2-ynylox...)
Affinity DataIC50:  9.90nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019618(1-(2-Allyloxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-y...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019614(1-(2-Butoxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-yl)...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019636(2-(4-Methyl-piperazin-1-yl)-1-(2-vinyloxy-ethyl)-1...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019607(1-(2-Ethoxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019629(1-(2-Ethoxy-ethyl)-2-piperazin-1-yl-1H-benzoimidaz...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019596(2-(4-Methyl-piperazin-1-yl)-1-(2-prop-2-ynyloxy-et...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM35938(1-(p-chlorophenyl)-1-(2-pyridyl)-3-N,N-dimethylpro...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019634(1-(2-Methoxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019597(2-(4-Butyl-piperazin-1-yl)-1-(2-ethoxy-ethyl)-1H-b...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019625(2-(4-Benzyl-[1,4]diazepan-1-yl)-1-(2-ethoxy-ethyl)...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019611(2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-propoxy-ethyl...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019631(1-(2-Ethoxy-ethyl)-2-(4-propyl-piperazin-1-yl)-1H-...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019630(1-(2-Ethoxy-ethyl)-2-(4-ethyl-[1,4]diazepan-1-yl)-...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019617(1-(2-Allyloxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1...)
Affinity DataIC50:  17nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019616(1-Benzyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimida...)
Affinity DataIC50:  17nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019619(2-(4-Methyl-piperazin-1-yl)-1-propoxymethyl-1H-ben...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019635(1-(2-Ethoxy-ethyl)-2-(4-ethyl-piperazin-1-yl)-1H-b...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019593(1-(2-Ethylsulfanyl-ethyl)-2-(4-methyl-piperazin-1-...)
Affinity DataIC50:  19nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019626(2-(4-Methyl-piperazin-1-yl)-1-pentyl-1H-benzoimida...)
Affinity DataIC50:  19nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019599(2-(4-Methyl-piperazin-1-yl)-1-(2-propoxy-ethyl)-1H...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019639(2-[1,4]Diazepan-1-yl-1-(2-ethoxy-ethyl)-1H-benzoim...)
Affinity DataIC50:  25nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019632(1-Hexyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidaz...)
Affinity DataIC50:  26nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019627(2-(4-Benzyl-piperazin-1-yl)-1-(2-ethoxy-ethyl)-1H-...)
Affinity DataIC50:  27nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019601(1-(2-Ethoxy-ethyl)-2-(4-pentyl-piperazin-1-yl)-1H-...)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019592(1-(2-Ethoxy-ethyl)-2-(4-phenethyl-piperazin-1-yl)-...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019613(1-(2-Butoxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-...)
Affinity DataIC50:  38nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019594(2-{2-[2-(4-Methyl-piperazin-1-yl)-benzoimidazol-1-...)
Affinity DataIC50:  42nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019620(1-Butyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidaz...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019633(2-(4-Methyl-piperazin-1-yl)-1-propylsulfanylmethyl...)
Affinity DataIC50:  68nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019598(1-Heptyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimida...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019610(2-(4-Methyl-piperazin-1-yl)-1-phenethyl-1H-benzoim...)
Affinity DataIC50:  240nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019608(CHEMBL17959 | Ethyl-{2-[2-(4-methyl-piperazin-1-yl...)
Affinity DataIC50:  290nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019622(1-Methyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimida...)
Affinity DataIC50:  320nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019606(2-(4-Methyl-piperazin-1-yl)-1-propyl-1H-benzoimida...)
Affinity DataIC50:  380nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019641(2-[2-(4-Methyl-piperazin-1-yl)-benzoimidazol-1-yl]...)
Affinity DataIC50:  410nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019637(1-(2-Benzyloxy-ethyl)-2-(4-methyl-piperazin-1-yl)-...)
Affinity DataIC50:  430nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019612(1-(2-Methyl-pentyl)-2-(4-methyl-piperazin-1-yl)-1H...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019603(1-(3-Ethylsulfanyl-propyl)-2-(4-methyl-piperazin-1...)
Affinity DataIC50:  530nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019642(2-(4-Methyl-piperazin-1-yl)-1-phenyl-1H-benzoimida...)
Affinity DataIC50:  760nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019600(1-(3-Methoxy-propyl)-2-(4-methyl-piperazin-1-yl)-1...)
Affinity DataIC50:  860nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019621(1-(1-Methyl-butyl)-2-(4-methyl-piperazin-1-yl)-1H-...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50019645(1-(3-Methyl-butyl)-2-(4-methyl-piperazin-1-yl)-1H-...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibition of histamine-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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