Compile Data Set for Download or QSAR
maximum 50k data
Found 47 Enz. Inhib. hit(s) with all data for entry = 50001685
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of KDR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of Ron (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  19nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  21nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  21nMAssay Description:Inhibition of KDR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  29nMAssay Description:Inhibition of [125I]VCAM-Ig binding to VLA-4 of Jurkat cells in the presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297565(CHEMBL4160512)
Affinity DataIC50:  30nMAssay Description:In vitro antiviral activity against HIV-1 Reverse transcriptase M184V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297346(CHEMBL4167741)
Affinity DataIC50:  37nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  37nMAssay Description:Inhibition of RET (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297285(CHEMBL4161786)
Affinity DataIC50:  46nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296469(CHEMBL4166652)
Affinity DataIC50:  50nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  53nMAssay Description:Inhibition of c-Kit (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  61nMAssay Description:Inhibition of Src (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297158(CHEMBL4175371)
Affinity DataIC50:  61nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  62nMAssay Description:Inhibition of AXL (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage-stimulating protein receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  69nMAssay Description:Inhibition of Ron (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296409(CHEMBL4163825)
Affinity DataIC50:  94nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297512(CHEMBL4174964)
Affinity DataIC50:  97nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297344(CHEMBL4175612)
Affinity DataIC50:  114nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  128nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297405(CHEMBL4168185)
Affinity DataIC50:  141nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  152nMAssay Description:Inhibition of RET (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296346(CHEMBL4172427)
Affinity DataIC50:  154nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296407(CHEMBL4160448)
Affinity DataIC50:  169nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  178nMAssay Description:Inhibition of [125I]VCAM-Ig binding to VLA-4 of Jurkat cells in the presence of Mn2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296471(CHEMBL4160268)
Affinity DataIC50:  196nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296399(CHEMBL4175433)
Affinity DataIC50:  205nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296750(CHEMBL4164749)
Affinity DataIC50:  308nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296402(CHEMBL4166841)
Affinity DataIC50:  320nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296398(CHEMBL4164120)
Affinity DataIC50:  331nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296470(CHEMBL4177280)
Affinity DataIC50:  337nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296408(CHEMBL4168353)
Affinity DataIC50:  348nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296404(CHEMBL4175145)
Affinity DataIC50:  358nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296403(CHEMBL4167282)
Affinity DataIC50:  415nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296401(CHEMBL4177459)
Affinity DataIC50:  427nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296405(CHEMBL4170667)
Affinity DataIC50:  495nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296410(CHEMBL4171699)
Affinity DataIC50:  580nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296406(CHEMBL4160024)
Affinity DataIC50:  658nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296400(CHEMBL4167564)
Affinity DataIC50:  659nMAssay Description:Inhibition of VLA-4 binding in Jurkat cells in the presence of Mg2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296397(CHEMBL4171989)
Affinity DataIC50:  688nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  812nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296349(CHEMBL4160329)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50296396(CHEMBL4170935)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50297394(CHEMBL4171115)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of IGF1R (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Zhuhai Campus Of Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of IGF1R (unknown origin) using poly (Glu,Tyr) 4:1 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed