Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50002882
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024694((S)-6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethy...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024698(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024687((+/-)-6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymet...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024688(9-Imidazol-1-yl-8-(4-methoxy-benzyloxymethyl)-non-...)
Affinity DataIC50:  390nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024685((R)-6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethy...)
Affinity DataIC50:  420nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50023002(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  540nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024693(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  560nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024684(5-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  730nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024691(5-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  750nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024699(9-Imidazol-1-yl-8-(4-methoxy-benzyloxymethyl)-nona...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM7962(4-(2-Imidazol-1-yl-ethoxy)-benzoic acid; hydrochlo...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024690(9-Imidazol-1-yl-8-(4-methoxy-benzyloxymethyl)-nona...)
Affinity DataIC50:  1.43E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024696(7-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024686(7-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024692(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  8.33E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024697(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024695(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Searle Research And Development

Curated by ChEMBL
LigandPNGBDBM50024689(8-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed