Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50029209
LigandPNGBDBM50282270(4'-(2-Butyl-4-cyclopentyl-4-methyl-5-oxo-4,5-dihyd...)
Affinity DataIC50:  3.30nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282264(2-Butyl-5-cyclohexyl-5-methyl-3-[2'-(1H-tetrazol-5...)
Affinity DataIC50:  5.20nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282264(2-Butyl-5-cyclohexyl-5-methyl-3-[2'-(1H-tetrazol-5...)
Affinity DataIC50:  5.20nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282267(4'-(2-Butyl-4-isopropyl-4-methyl-5-oxo-4,5-dihydro...)
Affinity DataIC50:  7.30nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282263(2-Butyl-5-cyclopentyl-5-methyl-3-[2'-(2H-tetrazol-...)
Affinity DataIC50:  7.60nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282262(4'-(2-Butyl-4-cyclohexyl-4-methyl-5-oxo-4,5-dihydr...)
Affinity DataIC50:  12nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282268(4'-(2-Butyl-4-cyclopropyl-4-methyl-5-oxo-4,5-dihyd...)
Affinity DataIC50:  18nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282265(4'-(2-Butyl-4-methyl-5-oxo-4-phenyl-4,5-dihydro-im...)
Affinity DataIC50:  19nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042244(4'-(2-Butyl-4,4-dimethyl-5-oxo-4,5-dihydro-imidazo...)
Affinity DataIC50:  35nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282269(4'-(2-Butyl-4-cyclohexyl-4-ethyl-5-oxo-4,5-dihydro...)
Affinity DataIC50:  52nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042240(4'-(2-Butyl-4,4-diethyl-5-oxo-4,5-dihydro-imidazol...)
Affinity DataIC50:  56nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042239(4'-(2-Butyl-4,4-dicyclopropyl-5-oxo-4,5-dihydro-im...)
Affinity DataIC50:  80nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282266(4'-(2-Butyl-4-cyclohexylmethyl-4-methyl-5-oxo-4,5-...)
Affinity DataIC50:  150nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282271(4'-[2-Butyl-4-(2,4-dimethyl-pentyl)-4-methyl-5-oxo...)
Affinity DataIC50:  230nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042222(4'-(2,4,4-Tributyl-5-oxo-4,5-dihydro-imidazol-1-yl...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50042241(4'-(2-Butyl-4,4-diisobutyl-5-oxo-4,5-dihydro-imida...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article