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Found 24 Enz. Inhib. hit(s) with all data for entry = 50029436
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50117909(CHEMBL278176 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284470(Benzo[1,3]dioxol-5-yl-[4-(2-ethyl-5,7-dimethyl-imi...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50117909(CHEMBL278176 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284468(5-Isobutyl-thiophene-2-sulfonic acid {2-benzo[1,3]...)
Affinity DataIC50:  75nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284468(5-Isobutyl-thiophene-2-sulfonic acid {2-benzo[1,3]...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284470(Benzo[1,3]dioxol-5-yl-[4-(2-ethyl-5,7-dimethyl-imi...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284472(CHEMBL15573 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-e...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284466(5-Isobutyl-3H-1lambda*4*-thiophene-2-sulfonic acid...)
Affinity DataIC50:  420nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284469(CHEMBL16197 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-e...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284474(3H-1lambda*4*-Thiophene-2-sulfonic acid {2-benzo[1...)
Affinity DataIC50:  540nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284466(5-Isobutyl-3H-1lambda*4*-thiophene-2-sulfonic acid...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284467(CHEMBL16018 | Propane-2-sulfonic acid {2-benzo[1,3...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284473(CHEMBL274243 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284474(3H-1lambda*4*-Thiophene-2-sulfonic acid {2-benzo[1...)
Affinity DataIC50:  820nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284471(Benzo[1,3]dioxol-5-yl-[4-(2-ethyl-5,7-dimethyl-imi...)
Affinity DataIC50:  840nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284469(CHEMBL16197 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-e...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284472(CHEMBL15573 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-e...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284471(Benzo[1,3]dioxol-5-yl-[4-(2-ethyl-5,7-dimethyl-imi...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284473(CHEMBL274243 | N-{2-Benzo[1,3]dioxol-5-yl-2-[4-(2-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284467(CHEMBL16018 | Propane-2-sulfonic acid {2-benzo[1,3...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175515((2,5-Dibromo-3,4-dimethoxy-phenyl)-[4-(2-ethyl-5,7...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284444(CHEMBL15689 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human endothelin A (ETA) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175515((2,5-Dibromo-3,4-dimethoxy-phenyl)-[4-(2-ethyl-5,7...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284444(CHEMBL15689 | [4-(2-Ethyl-5,7-dimethyl-imidazo[4,5...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of human endothelin B (ETB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article