Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50029554
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285512(CHEMBL77612 | N-{[(2,4,6-trimethoxyphenyl)amino]ca...)
Affinity DataIC50:  85nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285501(CHEMBL77898 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  86nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cholesterol fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285500(CHEMBL76780 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  520nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cholesterol fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285501(CHEMBL77898 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  675nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285511(CHEMBL433319 | N-{[(2,6-isopropylphenyl)amino]carb...)
Affinity DataIC50:  682nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285507(CHEMBL76251 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  830nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cholesterol fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285513(CHEMBL306626 | N-{[(2,6-isopropylphenyl)amino]carb...)
Affinity DataIC50:  830nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285507(CHEMBL76251 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  940nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285502(CHEMBL77583 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Compound at 5 microM concentration was tested in vitro for inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cho...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285504(CHEMBL420942 | N-{[(2,6-isopropylphenyl)amino]carb...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cholesterol fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285509(CHEMBL76037 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285510(CHEMBL75853 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285509(CHEMBL76037 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cholesterol fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285506(CHEMBL75975 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285504(CHEMBL420942 | N-{[(2,6-isopropylphenyl)amino]carb...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285498(CHEMBL309595 | N-{[(2,6-isopropylphenyl)amino]carb...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cholesterol fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285498(CHEMBL309595 | N-{[(2,6-isopropylphenyl)amino]carb...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285503(CHEMBL76088 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cholesterol fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285503(CHEMBL76088 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50040468(2,6-Bis(1-methylethyl)phenyl[[2,6-Bis(1-methylethy...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285497(CHEMBL430795 | N-{[(2,4,6-methoxyphenyl)amino]carb...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285499(CHEMBL76524 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  8.83E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285502(CHEMBL77583 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285505(CHEMBL75865 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in intestinal microsomes of cholesterol fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285505(CHEMBL75865 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  1.36E+4nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285508(CHEMBL77054 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  2.26E+4nMAssay Description:Inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of cholesterol fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSterol O-acyltransferase 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285500(CHEMBL76780 | N-{[(2,6-isopropylphenyl)amino]carbo...)
Affinity DataIC50:  3.80E+4nMAssay Description:Compound at 5 microM concentration was tested in vitro for inhibition of Acyl-CoA: Cholesterol Acyltransferase (ACAT) in liver microsomes of choleste...More data for this Ligand-Target Pair
In DepthDetails Article