Affinity DataKi: 12nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 131nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 229nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 428nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 551nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.28E+3nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibitory activity against Adenosine A1 receptor binding siteMore data for this Ligand-Target Pair
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibitory activity against Adenosine A2a receptor binding siteMore data for this Ligand-Target Pair