Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50029574
LigandPNGBDBM50285769(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285760(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285761(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285767(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.300nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285752(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.400nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285768(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50031530(2-Butyl-4-(methylthio)-1-[[2'-[[[(propylamino)carb...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285770(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285762(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285763(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.600nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285754(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.700nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285762(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.900nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285764(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285763(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285752(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285757(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285753(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285755(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.90nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285758(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285754(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285758(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285757(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2.80nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285771(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2.90nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285756(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.80nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285766(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.90nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285770(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.90nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285766(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  4.70nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285765(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  4.80nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285765(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  5nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285764(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  5.60nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285755(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  6.30nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285759(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  6.60nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285768(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  8nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285756(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  8.20nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285767(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  9.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285759(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285761(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  38nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285769(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  44nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285760(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  120nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50031530(2-Butyl-4-(methylthio)-1-[[2'-[[[(propylamino)carb...)
Affinity DataIC50:  920nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285771(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.50E+3nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285753(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.80E+3nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article