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Found 32 Enz. Inhib. hit(s) with all data for entry = 50030057
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290697(CHEMBL96879 | {2-[3-(3-Carbamimidoyl-phenyl)-5-(4-...)
Affinity DataKi:  18nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM17283((2S)-3-(7-carbamimidoylnaphthalen-2-yl)-2-(4-{[(3S...)
Affinity DataKi:  41nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  94nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290699(CHEMBL94761 | [3-(4-Carbamimidoyl-phenyl)-5-(3-car...)
Affinity DataKi:  117nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290692(CHEMBL433351 | [3-(3-Carbamimidoyl-phenyl)-5-(4-ca...)
Affinity DataKi:  143nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290690(CHEMBL93445 | [3-(3-Carbamimidoyl-phenyl)-5-(3-car...)
Affinity DataKi:  230nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290694(3-(3-Carbamimidoyl-phenyl)-4,5-dihydro-isoxazole-5...)
Affinity DataKi:  270nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290697(CHEMBL96879 | {2-[3-(3-Carbamimidoyl-phenyl)-5-(4-...)
Affinity DataKi:  420nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  480nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290693(CHEMBL317590 | N-(3-Carbamimidoyl-phenyl)-2-[3-(4-...)
Affinity DataKi:  510nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290694(3-(3-Carbamimidoyl-phenyl)-4,5-dihydro-isoxazole-5...)
Affinity DataKi:  700nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290690(CHEMBL93445 | [3-(3-Carbamimidoyl-phenyl)-5-(3-car...)
Affinity DataKi:  800nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290693(CHEMBL317590 | N-(3-Carbamimidoyl-phenyl)-2-[3-(4-...)
Affinity DataKi:  870nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290692(CHEMBL433351 | [3-(3-Carbamimidoyl-phenyl)-5-(4-ca...)
Affinity DataKi: >1.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290699(CHEMBL94761 | [3-(4-Carbamimidoyl-phenyl)-5-(3-car...)
Affinity DataKi: >1.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290695(CHEMBL94563 | N-(3-Carbamimidoyl-phenyl)-2-[3-(3-c...)
Affinity DataKi: >1.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290691(CHEMBL97842 | N-(4-Carbamimidoyl-phenyl)-2-[3-(3-c...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290698(CHEMBL94799 | N-(4-Carbamimidoyl-phenyl)-2-[3-(4-c...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290695(CHEMBL94563 | N-(3-Carbamimidoyl-phenyl)-2-[3-(3-c...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290693(CHEMBL317590 | N-(3-Carbamimidoyl-phenyl)-2-[3-(4-...)
Affinity DataKi:  2.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290698(CHEMBL94799 | N-(4-Carbamimidoyl-phenyl)-2-[3-(4-c...)
Affinity DataKi:  2.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290697(CHEMBL96879 | {2-[3-(3-Carbamimidoyl-phenyl)-5-(4-...)
Affinity DataKi:  3.10E+3nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290691(CHEMBL97842 | N-(4-Carbamimidoyl-phenyl)-2-[3-(3-c...)
Affinity DataKi:  1.11E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290695(CHEMBL94563 | N-(3-Carbamimidoyl-phenyl)-2-[3-(3-c...)
Affinity DataKi:  1.12E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290690(CHEMBL93445 | [3-(3-Carbamimidoyl-phenyl)-5-(3-car...)
Affinity DataKi:  1.18E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50066615((E,Z)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-o...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290699(CHEMBL94761 | [3-(4-Carbamimidoyl-phenyl)-5-(3-car...)
Affinity DataKi:  1.41E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290694(3-(3-Carbamimidoyl-phenyl)-4,5-dihydro-isoxazole-5...)
Affinity DataKi:  1.60E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  1.60E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290692(CHEMBL433351 | [3-(3-Carbamimidoyl-phenyl)-5-(4-ca...)
Affinity DataKi: >2.10E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50058875((S)-3-{2-[3-(4-Carbamimidoyl-phenyl)-4,5-dihydro-i...)
Affinity DataKi:  3.85E+4nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041220(1,2-bis(5-amidinobenzofuran-2-yl)ethane | 2-(2-{5-...)
Affinity DataKi:  5.70E+5nMAssay Description:The compound was evaluated for inhibitory activity against bovine Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article