Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50048616
LigandPNGBDBM50029051((-)-arterenol | (-)-noradrenaline | (-)-norepineph...)
Affinity DataIC50:  16nMAssay Description:Binding affinity against Alpha adrenergic receptor using [3H]dihydroergocryptine radioligand in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50029050((-)-(R)-epinephrine | (-)-3,4-dihydroxy-alpha-((me...)
Affinity DataIC50:  17nMAssay Description:Binding affinity against Alpha adrenergic receptor using [3H]dihydroergocryptine radioligand in rat brain homogenateMore data for this Ligand-Target Pair
LigandPNGBDBM50223423(CHEMBL22352)
Affinity DataIC50:  4.00E+3nMAssay Description:Binding affinity against Alpha adrenergic receptor using [3H]dihydroergocryptine radioligand in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223424(CHEMBL280151)
Affinity DataIC50:  9.00E+3nMAssay Description:Binding affinity against Beta adrenergic receptor using [3H]dihydroalprenolol radioligand in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223422(CHEMBL22195)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity against Alpha adrenergic receptor using [3H]dihydroergocryptine radioligand in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50029050((-)-(R)-epinephrine | (-)-3,4-dihydroxy-alpha-((me...)
Affinity DataIC50:  2.90E+4nMAssay Description:Binding affinity against Beta adrenergic receptor using [3H]dihydroalprenolol radioligand in rat brain homogenateMore data for this Ligand-Target Pair
LigandPNGBDBM50223424(CHEMBL280151)
Affinity DataIC50:  3.30E+4nMAssay Description:Binding affinity against Alpha adrenergic receptor using [3H]dihydroergocryptine radioligand in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223422(CHEMBL22195)
Affinity DataIC50:  1.10E+5nMAssay Description:Binding affinity against Beta adrenergic receptor using [3H]dihydroalprenolol radioligand in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223423(CHEMBL22352)
Affinity DataIC50:  1.30E+5nMAssay Description:Binding affinity against Beta adrenergic receptor using [3H]dihydroalprenolol radioligand in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed