Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50036273
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKd:  1.5nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030081(CHEMBL265017 | [Mca1,D-Phe2,Sar7]AVP)
Affinity DataKd:  98nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030080(CHEMBL411420 | [Mca1,D-Tyr(OEt)2,Sar7]AVT)
Affinity DataKd:  130nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50368886(CHEMBL1793955)
Affinity DataKd:  265nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030083(CHEMBL414582 | [Mca1,D-Phe2,Sar7]AVT)
Affinity DataKd:  311nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030077(CHEMBL330022 | [Mca1,D-Tyr(OMe)2,Sar7]AVT)
Affinity DataKd:  18nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030087(CHEMBL274397 | [Mca1,D-Trp2,Sar7]AVT)
Affinity DataKd:  6nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030086(CHEMBL265264 | [Mca1,Sar7]AVP)
Affinity DataKd:  240nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030085(CHEMBL415230 | [Mpa1,D-Tyr(OEt)2,Sar7]AVT)
Affinity DataKd:  27nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030083(CHEMBL414582 | [Mca1,D-Phe2,Sar7]AVT)
Affinity DataKd:  8nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030081(CHEMBL265017 | [Mca1,D-Phe2,Sar7]AVP)
Affinity DataKd:  7nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030085(CHEMBL415230 | [Mpa1,D-Tyr(OEt)2,Sar7]AVT)
Affinity DataKd:  35nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030088(CHEMBL438387 | [Mca1,D-Tyr(OEt)2,Sar7]AVP)
Affinity DataKd:  29nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030079(CHEMBL87636 | [Mpa1,D-Phe2,Sar7]AVT)
Affinity DataKd:  421nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030077(CHEMBL330022 | [Mca1,D-Tyr(OMe)2,Sar7]AVT)
Affinity DataKd:  811nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030079(CHEMBL87636 | [Mpa1,D-Phe2,Sar7]AVT)
Affinity DataKd:  8nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030080(CHEMBL411420 | [Mca1,D-Tyr(OEt)2,Sar7]AVT)
Affinity DataKd:  15nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030089(CHEMBL384292 | [Mca1,D-Tyr2,Sar7]AVP)
Affinity DataKd:  160nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030089(CHEMBL384292 | [Mca1,D-Tyr2,Sar7]AVP)
Affinity DataKd:  230nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030087(CHEMBL274397 | [Mca1,D-Trp2,Sar7]AVT)
Affinity DataKd:  3.00E+5nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50030088(CHEMBL438387 | [Mca1,D-Tyr(OEt)2,Sar7]AVP)
Affinity DataKd:  21nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50368886(CHEMBL1793955)
Affinity DataKd:  182nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Max-Planck-Institut F£R Biophysik

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKd:  6.70nMAssay Description:Inhibition of radioligand [3H]OT binding to oxytocin receptor (OT) in guinea pig myometrium membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed