Compile Data Set for Download or QSAR
maximum 50k data
Found 43 Enz. Inhib. hit(s) with all data for entry = 50036356
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033236(8,9-Dichloro-2-methyl-5-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50:  0.300nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033242(3-Cyclohexyl-6-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.400nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033257(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033240(1-Methyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  0.600nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033238(3-(4-Chloro-phenyl)-1,8-dimethyl-5-[4-(2-methyl-im...)
Affinity DataIC50:  0.600nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033264(3-Cyclohexyl-1,8-dimethyl-5-[4-(2-methyl-imidazo[4...)
Affinity DataIC50:  0.700nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033260(3-Isobutoxymethyl-1,8-dimethyl-5-[4-(2-methyl-imid...)
Affinity DataIC50:  0.800nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033234(1,3-Dimethyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033233(8,9-Dichloro-1-methyl-5-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50:  1.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033249(5,7,9-Trimethyl-2-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  1.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033229(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033245(8-Bromo-5-methyl-2-[4-(2-methyl-imidazo[4,5-c]pyri...)
Affinity DataIC50:  1.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033255(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033232(8,9-Dichloro-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1.70nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033263(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  2.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033231(1,8,9-Trimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  2.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033251(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  2.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033246(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  2.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033243(1-Methyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  2.70nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033230(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  3.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033241(3-Isopropyl-1,8-dimethyl-5-[4-(2-methyl-imidazo[4,...)
Affinity DataIC50:  3.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033268(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  3.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033235(7-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033254(8-Bromo-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl)...)
Affinity DataIC50:  4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033239(8-Bromo-1-methyl-4-[4-(2-methyl-imidazo[4,5-c]pyri...)
Affinity DataIC50:  4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)
Affinity DataIC50:  4.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033266(1,3,4-Trimethyl-7-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033237(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  5.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033267(8-Bromo-4-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl)...)
Affinity DataIC50:  5.60nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033253(3-(2-Methoxy-ethoxymethyl)-1,8-dimethyl-5-[4-(2-me...)
Affinity DataIC50:  6.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033258(7,9-Dimethyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  6.80nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033248(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  11nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033256(3-Hydroxymethyl-1,8-dimethyl-5-[4-(2-methyl-imidaz...)
Affinity DataIC50:  14nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033261(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  14nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033228(1,3,8-Trimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  17nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033227(7,9-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  21nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033262(1,3-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  26nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033247(1,7,9-Trimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  38nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033252(1-Methyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  45nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033244(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  55nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033265(4-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  66nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50038755(6-(2-chlorophenyl)-1-methyl-8,9-dihydro-4H,7H-cycl...)
Affinity DataIC50:  73nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033259(2-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  130nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed