Compile Data Set for Download or QSAR
maximum 50k data
Found 115 Enz. Inhib. hit(s) with all data for entry = 50005371
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50010096(CHEMBL12980 | Hydroxy-diphenyl-acetic acid 1-aza-b...)
Affinity DataKi:  0.0450nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50010096(CHEMBL12980 | Hydroxy-diphenyl-acetic acid 1-aza-b...)
Affinity DataKi:  0.0510nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50010096(CHEMBL12980 | Hydroxy-diphenyl-acetic acid 1-aza-b...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036185(3-(2'-Benzofuranyl)-quinuclidine-2-ene | 3-Benzofu...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  14nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036185(3-(2'-Benzofuranyl)-quinuclidine-2-ene | 3-Benzofu...)
Affinity DataKi:  31nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036195(3-Benzofuran-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene | ...)
Affinity DataKi:  34nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036173(3-Benzo[b]thiophen-3-yl-1-aza-bicyclo[2.2.2]oct-2-...)
Affinity DataKi:  37nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036171(3-Benzofuran-2-yl-1-aza-bicyclo[2.2.2]octane | CHE...)
Affinity DataKi:  57nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036175(3-(2,3-Dihydro-benzofuran-2-yl)-1-aza-bicyclo[2.2....)
Affinity DataKi:  59nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036185(3-(2'-Benzofuranyl)-quinuclidine-2-ene | 3-Benzofu...)
Affinity DataKi:  59nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036175(3-(2,3-Dihydro-benzofuran-2-yl)-1-aza-bicyclo[2.2....)
Affinity DataKi:  59nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036183(3-(2'-Benzothiophenyl)-quinuclidine-2-ene | 3-Benz...)
Affinity DataKi:  81nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036173(3-Benzo[b]thiophen-3-yl-1-aza-bicyclo[2.2.2]oct-2-...)
Affinity DataKi:  96nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036195(3-Benzofuran-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene | ...)
Affinity DataKi:  99nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036190(3-Benzooxazol-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene |...)
Affinity DataKi:  100nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  110nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036173(3-Benzo[b]thiophen-3-yl-1-aza-bicyclo[2.2.2]oct-2-...)
Affinity DataKi:  110nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036195(3-Benzofuran-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene | ...)
Affinity DataKi:  160nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036175(3-(2,3-Dihydro-benzofuran-2-yl)-1-aza-bicyclo[2.2....)
Affinity DataKi:  160nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036175(3-(2,3-Dihydro-benzofuran-2-yl)-1-aza-bicyclo[2.2....)
Affinity DataKi:  160nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036170(3-Benzothiazol-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene ...)
Affinity DataKi:  170nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036171(3-Benzofuran-2-yl-1-aza-bicyclo[2.2.2]octane | CHE...)
Affinity DataKi:  200nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036193(3-(2-Methoxy-phenyl)-1-aza-bicyclo[2.2.2]oct-2-ene...)
Affinity DataKi:  220nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036171(3-Benzofuran-2-yl-1-aza-bicyclo[2.2.2]octane | CHE...)
Affinity DataKi:  240nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036183(3-(2'-Benzothiophenyl)-quinuclidine-2-ene | 3-Benz...)
Affinity DataKi:  270nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  270nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036182(3-Thiophen-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene | CH...)
Affinity DataKi:  290nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036196(3-Furan-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene | CHEMB...)
Affinity DataKi:  300nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036194(2-(1-Aza-bicyclo[2.2.2]oct-2-en-3-yl)-phenol | CHE...)
Affinity DataKi:  330nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036175(3-(2,3-Dihydro-benzofuran-2-yl)-1-aza-bicyclo[2.2....)
Affinity DataKi:  340nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036194(2-(1-Aza-bicyclo[2.2.2]oct-2-en-3-yl)-phenol | CHE...)
Affinity DataKi:  360nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036163(3-Benzofuran-2-yl-1-methyl-1-azonia-bicyclo[2.2.2]...)
Affinity DataKi:  360nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036196(3-Furan-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene | CHEMB...)
Affinity DataKi:  390nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036190(3-Benzooxazol-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene |...)
Affinity DataKi:  400nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036169(3-Selenophen-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene | ...)
Affinity DataKi:  410nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036193(3-(2-Methoxy-phenyl)-1-aza-bicyclo[2.2.2]oct-2-ene...)
Affinity DataKi:  410nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036183(3-(2'-Benzothiophenyl)-quinuclidine-2-ene | 3-Benz...)
Affinity DataKi:  420nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036163(3-Benzofuran-2-yl-1-methyl-1-azonia-bicyclo[2.2.2]...)
Affinity DataKi:  460nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036192(3-Benzofuran-2-yl-1-methyl-1-azonia-bicyclo[2.2.2]...)
Affinity DataKi:  520nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036191(3-Furan-2-yl-1-aza-bicyclo[2.2.2]octane | CHEMBL14...)
Affinity DataKi:  540nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036170(3-Benzothiazol-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene ...)
Affinity DataKi:  600nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036182(3-Thiophen-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene | CH...)
Affinity DataKi:  620nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036165(3-Thiophen-3-yl-1-aza-bicyclo[2.2.2]oct-2-ene | CH...)
Affinity DataKi:  710nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036190(3-Benzooxazol-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene |...)
Affinity DataKi:  720nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036193(3-(2-Methoxy-phenyl)-1-aza-bicyclo[2.2.2]oct-2-ene...)
Affinity DataKi:  740nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036177(3-Benzofuran-2-yl-1-aza-bicyclo[2.2.2]octan-3-ol |...)
Affinity DataKi:  810nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036186(3-Benzo[b]thiophen-3-yl-1-aza-bicyclo[2.2.2]octan-...)
Affinity DataKi:  820nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036169(3-Selenophen-2-yl-1-aza-bicyclo[2.2.2]oct-2-ene | ...)
Affinity DataKi:  990nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50036180(3-Benzo[b]thiophen-2-yl-1-aza-bicyclo[2.2.2]octan-...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M1 by measuring displacement of [3H]-QNB from guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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