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Found 32 Enz. Inhib. hit(s) with all data for entry = 50036298
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368929(CHEMBL610155)
Affinity DataKi:  7nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453502(CHEMBL2113573)
Affinity DataKi:  7.5nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453499(CHEMBL2113598)
Affinity DataKi:  7.90nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368937(CHEMBL609252)
Affinity DataKi:  8.30nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453507(CHEMBL2113584)
Affinity DataKi:  11nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368922(CHEMBL611311)
Affinity DataKi:  14nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368950(CHEMBL610442)
Affinity DataKi:  14nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453512(CHEMBL2113599)
Affinity DataKi:  23nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453510(CHEMBL2113586)
Affinity DataKi:  26nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453511(CHEMBL2113587)
Affinity DataKi:  29nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368930(CHEMBL607875)
Affinity DataKi:  39nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368940(CHEMBL611000)
Affinity DataKi:  39nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368928(CHEMBL611600)
Affinity DataKi:  50nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368931(CHEMBL608964)
Affinity DataKi:  50nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453500(CHEMBL2113596)
Affinity DataKi:  62nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453508(CHEMBL2113585)
Affinity DataKi:  110nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453501(CHEMBL2113597)
Affinity DataKi:  120nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368952(CHEMBL610717)
Affinity DataKi:  130nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368939(CHEMBL611598)
Affinity DataKi:  140nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368941(CHEMBL608369)
Affinity DataKi:  140nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453505(CHEMBL2113589)
Affinity DataKi:  150nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368951(CHEMBL611599)
Affinity DataKi:  160nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368943(CHEMBL609554)
Affinity DataKi:  160nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368953(CHEMBL608962)
Affinity DataKi:  170nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368947(CHEMBL610724)
Affinity DataKi:  170nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50368927(CHEMBL609555)
Affinity DataKi:  180nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453504(CHEMBL2113591)
Affinity DataKi:  200nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453498(CHEMBL2113594)
Affinity DataKi:  370nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453509(CHEMBL2113603)
Affinity DataKi:  510nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453513(CHEMBL2113579)
Affinity DataKi:  890nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453503(CHEMBL2113590)
Affinity DataKi:  895nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Carpibem

Curated by ChEMBL
LigandPNGBDBM50453506(CHEMBL2113583)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed