Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50005654
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039364(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039376(CHEMBL80773 | {5-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039345(CHEMBL77783 | Methyl-{5-methyl-7-propyl-8-[2'-(1H-...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039366(2-(2-Hydroxy-ethyl)-5-methyl-7-propyl-8-[2'-(1H-te...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039344(2-Ethyl-5-methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039372(CHEMBL80380 | {5-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039341(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039378(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039362(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039350(5-Hydroxymethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039346(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039374(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039357(CHEMBL312632 | {5-Methyl-3-oxo-7-propyl-8-[2'-(1H-...)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039347(2-Methoxymethyl-5-methyl-7-propyl-8-[2'-(1H-tetraz...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039368(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039342(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039370(2-Methoxy-5-methyl-7-propyl-8-[2'-(1H-tetrazol-5-y...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039371(CHEMBL76149 | {2-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039351(7-Butyl-5-methyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039352(CHEMBL80967 | {5-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039369(2,5-Dimethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039365(7-Ethyl-5-methyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039339(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039348(2-[4-(5-Methyl-3-oxo-7-propyl-2,3-dihydro-[1,2,4]t...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039375(7-Propyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataKi:  46nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039354(7-Propyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039361(2,5-Dimethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataKi:  53nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039358(7-Cyclopropyl-5-methyl-8-[2'-(1H-tetrazol-5-yl)-bi...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039379(5-Methoxymethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataKi:  92nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039363(CHEMBL80161 | {5-Methyl-7-propyl-8-[2'-(1H-tetrazo...)
Affinity DataKi:  99nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039373(7-Butyl-5-methyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  106nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039343(5-Methoxymethyl-2-methyl-7-propyl-8-[2'-(1H-tetraz...)
Affinity DataKi:  111nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039355(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  127nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039349(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  139nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039360(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  147nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039340(5-Methyl-2-methylsulfanyl-7-propyl-8-[2'-(1H-tetra...)
Affinity DataKi:  174nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039359(5-Methyl-2-phenyl-7-propyl-8-[2'-(1H-tetrazol-5-yl...)
Affinity DataKi:  175nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039367(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  185nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039353(5-Ethyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  225nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039380(4'-(7-Butyl-2-hydroxy-5-methyl-[1,2,4]triazolo[1,5...)
Affinity DataKi:  622nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039356(5,7-Dipropyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl-4-y...)
Affinity DataKi:  659nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039377(5-Methylsulfanyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Carpibem

Curated by ChEMBL
LigandPNGBDBM50039342(5-Methyl-7-propyl-8-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataKi:  7.92E+4nMAssay Description:In vitro binding affinitity against angiotensin-2 (AT-2) receptor in rat adrenalMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed