Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50007095
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058204((S)-2-{[6-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058199((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058202((S)-2-[(2-{(S)-2-[((R)-2-Amino-3-mercapto-propiony...)
Affinity DataIC50:  5nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058208((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058200((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  17nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058204((S)-2-{[6-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  17.5nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ki-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)
Affinity DataIC50:  37nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058195((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  44nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058198((S)-2-{[5-((R)-2-Amino-3-mercapto-propionylamino)-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058197((S)-2-{[6-((R)-2-Amino-3-mercapto-propionylamino)-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058193((S)-2-{[6-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  80nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058207((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  210nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058196((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  325nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058193((S)-2-{[6-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  500nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ki-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058205((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  950nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058197((S)-2-{[6-((R)-2-Amino-3-mercapto-propionylamino)-...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ki-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058206((S)-2-({(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propi...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058203((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  2.22E+3nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058194((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-nap...)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Centre De Recherches De Vitry-Alfortville

Curated by ChEMBL
LigandPNGBDBM50058201((S)-2-{(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propio...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of [3H]-FPP incorporation into human Ha-Ras by farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed