Affinity DataKi: 0.340nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by DAMGO (Opioid receptor mu 1)More data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Binding affinity against Opioid receptor mu 1 using [3H]naloxone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by DAMGO (Opioid receptor mu 1)More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by U69,593 in Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding activity against Opioid receptor mu 1 using [3H]-DAMGO as radioligand in rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity against Opioid receptor mu 1 using [3H]-Naloxone as radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by U69,593 in Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding activity against Opioid receptor mu 1 using [3H]-DAMGO as radioligand in rat brain membranes.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Binding affinity against Opioid receptor kappa 1 using [3H]ethylketocyclazocine as radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Binding activity against Opioid receptor kappa 1 using [3H]U69,593 as radioligand in guinea pig membranes .More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1)More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding activity against kOpioid receptor kappa 1 using [3H]U69,593 as radioligand in guinea pig membranes .More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1)More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by DAMGO (Opioid receptor mu 1)More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity against Opioid receptor kappa 1 using [3H]-Ethylketocyclazocine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity against Opioid receptor mu 1 using [3H]-Naloxone as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Binding activity against Opioid receptor delta 1 using [3H]-DADLE as radioligand in rat brain membranes.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 105nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by U69,593 in Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 166nMAssay Description:Binding activity against Opioid receptor mu 1 using [3H]-DAMGO as radioligand in rat brain membranes.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 272nMAssay Description:Binding activity against Opioid receptor delta 1 using [3H]-DADLE as radioligand in rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Inhibition of [35S]-GTP-gammaS, binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1)More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: 816nMAssay Description:Binding activity against Opioid receptor kappa 1 using [3H]U69,593 as radioligand in guinea pig membranes .More data for this Ligand-Target Pair
Affinity DataKi: 833nMAssay Description:Binding affinity against Opioid receptor kappa 1 using [3H]-Ethylketocyclazocine as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding activity against Opioid receptor delta 1 using [3H]-DADLE as radioligand in rat brain membranes.More data for this Ligand-Target Pair