Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50008043
TargetProthrombin(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50070307((1R,2S)-2-(2-Methylamino-3-naphthalen-2-yl-propion...)
Affinity DataIC50:  22nMAssay Description:Compound was evaluated for the inhibition of thrombin using the synthetic substrate chromozym THMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50228863((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50:  46nMAssay Description:Compound was evaluated for the inhibition of thrombin using the synthetic substrate chromozym THMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50070306((1R,2R)-2-(2-Methylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Compound was evaluated for the inhibition of thrombin using the synthetic substrate chromozym THMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50070305((1R,2S)-Cyclohexane-1,2-dicarboxylic acid 1-[((R)-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Compound was evaluated for the inhibition of thrombin using the synthetic substrate chromozym THMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50070304(CHEMBL281784 | Cyclohexane-1,2-dicarboxylic acid 1...)
Affinity DataIC50:  8.40E+4nMAssay Description:Compound was evaluated for the inhibition of thrombin using the synthetic substrate chromozym THMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed