BindingDB PrimarySearch

Found 27 Enz. Inhib. hit(s) with all data for entry = 50008199

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM17284(2-{[2-(5-carbamimidoyl-2-hydroxyphenoxy)-3,5-diflu...)

Ki: 0.110nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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PDB

3D Structure (crystal)

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50066623(CHEMBL72318 | {[2-(5-Carbamimidoyl-2-hydroxy-pheno...)

Ki: 0.410nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents

Details Article PubMed

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071415(3-[9-Benzyl-6-(5-carbamimidoyl-2-hydroxy-phenoxy)-...)

Ki: 0.420nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM17277((Z,Z)BABCH | 4-{[(1Z,3Z)-3-[(4-carbamimidoylphenyl...)

Ki: 0.660nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071419(3-[9-Benzyl-2-(5-carbamimidoyl-2-hydroxy-phenoxy)-...)

Ki: 10nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071417(3-[4-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-5,6...)

Ki: 19nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM17277((Z,Z)BABCH | 4-{[(1Z,3Z)-3-[(4-carbamimidoylphenyl...)

Ki: 30nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

CHEMBL MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed MMDB
PDB

3D Structure (crystal)

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50066633(3-[6-(3-Carbamimidoyl-phenoxy)-3,5-difluoro-4-meth...)

Ki: 80nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071418(3-[2-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-5,6...)

Ki: 81nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Coagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071416(3-[2-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-6,7...)

Ki: 106nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid

Details Article PubMed

Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM50071415(3-[9-Benzyl-6-(5-carbamimidoyl-2-hydroxy-phenoxy)-...)

Ki: 150nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM17284(2-{[2-(5-carbamimidoyl-2-hydroxyphenoxy)-3,5-diflu...)

Ki: 280nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

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Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM50071417(3-[4-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-5,6...)

Ki: 320nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM17277((Z,Z)BABCH | 4-{[(1Z,3Z)-3-[(4-carbamimidoylphenyl...)

Ki: 430nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071415(3-[9-Benzyl-6-(5-carbamimidoyl-2-hydroxy-phenoxy)-...)

Ki: 710nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM50071419(3-[9-Benzyl-2-(5-carbamimidoyl-2-hydroxy-phenoxy)-...)

Ki: 760nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071417(3-[4-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-5,6...)

Ki: 1.00E+3nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM50066623(CHEMBL72318 | {[2-(5-Carbamimidoyl-2-hydroxy-pheno...)

Ki: 1.10E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

CHEMBL PC cid PC sid Patents

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071419(3-[9-Benzyl-2-(5-carbamimidoyl-2-hydroxy-phenoxy)-...)

Ki: 1.30E+3nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM17284(2-{[2-(5-carbamimidoyl-2-hydroxyphenoxy)-3,5-diflu...)

Ki: 2.00E+3nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Purchase CHEMBL MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed

Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM50071418(3-[2-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-5,6...)

Ki: 2.20E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM50066633(3-[6-(3-Carbamimidoyl-phenoxy)-3,5-difluoro-4-meth...)

Ki: 2.70E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50066623(CHEMBL72318 | {[2-(5-Carbamimidoyl-2-hydroxy-pheno...)

Ki: 4.50E+3nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents

Details Article PubMed

Serine protease 1(Bos taurus (bovine))
Berlex Biosciences

Curated by ChEMBL

BDBM50071416(3-[2-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-6,7...)

Ki: >5.00E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

CHEMBL PC cid PC sid

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50066633(3-[6-(3-Carbamimidoyl-phenoxy)-3,5-difluoro-4-meth...)

Ki: >5.00E+3nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071418(3-[2-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-5,6...)

Ki: >5.00E+3nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Prothrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL

BDBM50071416(3-[2-(5-Carbamimidoyl-2-hydroxy-phenoxy)-6-oxo-6,7...)

Ki: >5.00E+3nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

CHEMBL PC cid PC sid

Details Article PubMed