TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 0.510nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low agonist state in rat striatal membranes using [3H]...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Affinity of compound for the D2 receptors in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [3H]-spip...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 45.8nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 258nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: >400nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 403nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 591nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 871nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair