Compile Data Set for Download or QSAR
maximum 50k data
Found 45 Enz. Inhib. hit(s) with all data for entry = 50008255
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071855(4-(4-Benzyl-piperazin-1-yl)-2-trifluoromethyl-1H-b...)
Affinity DataKi:  0.510nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071856(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-indol-2-on...)
Affinity DataKi:  0.560nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071858(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1H-indole | C...)
Affinity DataKi:  1.70nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071853(4-(4-Benzyl-piperazin-1-yl)-7-bromo-1H-indole | CH...)
Affinity DataKi:  2.60nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071855(4-(4-Benzyl-piperazin-1-yl)-2-trifluoromethyl-1H-b...)
Affinity DataKi:  2.90nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071856(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-indol-2-on...)
Affinity DataKi:  3nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  3.20nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071855(4-(4-Benzyl-piperazin-1-yl)-2-trifluoromethyl-1H-b...)
Affinity DataKi:  3.30nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low agonist state in rat striatal membranes using [3H]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071855(4-(4-Benzyl-piperazin-1-yl)-2-trifluoromethyl-1H-b...)
Affinity DataKi:  4.10nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071856(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-indol-2-on...)
Affinity DataKi:  5.40nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50069907(1-benzyl-4-(3-hydroxyphenyl)piperazine | 3-(4-Benz...)
Affinity DataKi:  5.5nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071856(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-indol-2-on...)
Affinity DataKi:  8nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071856(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-indol-2-on...)
Affinity DataKi:  8.10nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071859(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1,3-dihydro-i...)
Affinity DataKi:  8.80nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071858(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1H-indole | C...)
Affinity DataKi:  9.10nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071853(4-(4-Benzyl-piperazin-1-yl)-7-bromo-1H-indole | CH...)
Affinity DataKi:  12nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071854(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-benzoimida...)
Affinity DataKi:  14nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071855(4-(4-Benzyl-piperazin-1-yl)-2-trifluoromethyl-1H-b...)
Affinity DataKi:  15nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  15nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  17nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071853(4-(4-Benzyl-piperazin-1-yl)-7-bromo-1H-indole | CH...)
Affinity DataKi:  27nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50069907(1-benzyl-4-(3-hydroxyphenyl)piperazine | 3-(4-Benz...)
Affinity DataKi:  29nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  35nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071858(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1H-indole | C...)
Affinity DataKi:  42nMAssay Description:Affinity of compound for the D2 receptors in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [3H]-spip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071854(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-benzoimida...)
Affinity DataKi:  45.8nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071854(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-benzoimida...)
Affinity DataKi:  46nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071853(4-(4-Benzyl-piperazin-1-yl)-7-bromo-1H-indole | CH...)
Affinity DataKi:  47nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071852(4-(4-Benzyl-piperazin-1-yl)-1H-benzoimidazole | CH...)
Affinity DataKi:  47nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  53nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071853(4-(4-Benzyl-piperazin-1-yl)-7-bromo-1H-indole | CH...)
Affinity DataKi:  56nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071854(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-benzoimida...)
Affinity DataKi:  57nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071858(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1H-indole | C...)
Affinity DataKi:  81nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071859(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1,3-dihydro-i...)
Affinity DataKi:  85nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071854(4-(4-Benzyl-piperazin-1-yl)-1,3-dihydro-benzoimida...)
Affinity DataKi:  87nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071858(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1H-indole | C...)
Affinity DataKi:  95nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50069907(1-benzyl-4-(3-hydroxyphenyl)piperazine | 3-(4-Benz...)
Affinity DataKi:  95nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071852(4-(4-Benzyl-piperazin-1-yl)-1H-benzoimidazole | CH...)
Affinity DataKi:  107nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071852(4-(4-Benzyl-piperazin-1-yl)-1H-benzoimidazole | CH...)
Affinity DataKi:  107nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50069907(1-benzyl-4-(3-hydroxyphenyl)piperazine | 3-(4-Benz...)
Affinity DataKi:  246nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071852(4-(4-Benzyl-piperazin-1-yl)-1H-benzoimidazole | CH...)
Affinity DataKi:  258nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50069907(1-benzyl-4-(3-hydroxyphenyl)piperazine | 3-(4-Benz...)
Affinity DataKi: >400nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071859(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1,3-dihydro-i...)
Affinity DataKi:  403nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071859(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1,3-dihydro-i...)
Affinity DataKi:  540nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071859(4-(4-Benzyl-piperazin-1-yl)-5-chloro-1,3-dihydro-i...)
Affinity DataKi:  591nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071852(4-(4-Benzyl-piperazin-1-yl)-1H-benzoimidazole | CH...)
Affinity DataKi:  871nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed