Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 5877
TargetProthrombin(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM98168(US8487111, 8)
Affinity DataIC50:  16nMAssay Description:Thrombin inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCoagulation factor X(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM98166(US8487111, 2)
Affinity DataIC50:  21nMAssay Description:Factor Xa inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCoagulation factor X(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM98169(US8487111, 10)
Affinity DataIC50:  40nMAssay Description:Factor Xa inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCoagulation factor X(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM98167(US8487111, 6)
Affinity DataIC50:  70nMAssay Description:Factor Xa inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProthrombin(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM98169(US8487111, 10)
Affinity DataIC50:  74nMAssay Description:Thrombin inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCoagulation factor X(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM98168(US8487111, 8)
Affinity DataIC50:  167nMAssay Description:Factor Xa inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProthrombin(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM98167(US8487111, 6)
Affinity DataIC50:  186nMAssay Description:Thrombin inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProthrombin(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM98166(US8487111, 2)
Affinity DataIC50:  198nMAssay Description:Thrombin inhibitory activity.More data for this Ligand-Target Pair
In DepthDetails US Patent