Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50009266
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081724((4-{5-[1-Aza-bicyclo[2.2.2]oct-(3Z)-ylidenemethyl]...)
Affinity DataIC50: >10nMAssay Description:The compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081729(4-{5-[1-Aza-bicyclo[2.2.2]oct-(3Z)-ylidenemethyl]-...)
Affinity DataIC50: >10nMAssay Description:The compound was tested for its binding affinity against nicotinic receptor in synaptic membrane fractions from rat cerebral cortices.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081733(3-(3-Methyl-isoxazol-5-ylmethylene)-1-aza-bicyclo[...)
Affinity DataIC50:  12nMAssay Description:Compound was tested for its binding affinity against nicotinic receptor in synaptic membrane fractions from rat cerebral cortices.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50:  16nMAssay Description:Compound was tested for its binding affinity against nicotinic receptor in synaptic membrane fractions from rat cerebral cortices.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081734(3-[1-{3-[3,4-Bis-(4-methoxy-benzyloxy)-phenyl]-iso...)
Affinity DataIC50:  114nMAssay Description:The compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataIC50:  119nMAssay Description:Compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081731(3-[1-{3-[3,4-Bis-(4-methoxy-benzyloxy)-phenyl]-iso...)
Affinity DataIC50:  247nMAssay Description:The compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081728(3-[1-{3-[4-(4-Methoxy-benzyloxy)-phenyl]-isoxazol-...)
Affinity DataIC50:  250nMAssay Description:The compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081725(3-[1-{3-[3,4-Bis-(4-methoxy-benzyloxy)-phenyl]-iso...)
Affinity DataIC50:  260nMAssay Description:The compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081737(4-{5-[1-Aza-bicyclo[2.2.2]oct-(3E)-ylidenemethyl]-...)
Affinity DataIC50:  695nMAssay Description:The compound was tested for its binding affinity against nicotinic receptor in synaptic membrane fractions from rat cerebral cortices.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081735(4-{5-[1-Aza-bicyclo[2.2.2]oct-(3E)-ylidenemethyl]-...)
Affinity DataIC50:  803nMAssay Description:The compound was tested for its binding affinity against nicotinic receptor in synaptic membrane fractions from rat cerebral cortices.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081732((4-{5-[1-Aza-bicyclo[2.2.2]oct-(3E)-ylidenemethyl]...)
Affinity DataIC50:  806nMAssay Description:The compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081736(3-[1-{3-[4-(4-Methoxy-benzyloxy)-phenyl]-isoxazol-...)
Affinity DataIC50:  809nMAssay Description:The compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50081730(3-[1-{3-[3,4-Bis-(4-methoxy-benzyloxy)-phenyl]-iso...)
Affinity DataIC50:  1.23E+3nMAssay Description:The compound was tested for its binding affinity against M1 human recombinant muscarinic receptor in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed