Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 5299
TargetNociceptin receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM50083230(1-((3R,4R)-1-Cyclooctylmethyl-3-hydroxymethyl-pipe...)
Affinity DataKi:  1.51nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM50087016(8-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5...)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM85748(H-PHE-(R)-GLY-GLY-PHE-THR-GLY-ALA-ARG-LYS-SER-ALA-...)
Affinity DataKi:  4.27nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM85749(III-BTD | NOCICEPTIN RECEPTOR ANTAGONIST PEPTIDE I...)
Affinity DataKi:  8.91nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM85749(III-BTD | NOCICEPTIN RECEPTOR ANTAGONIST PEPTIDE I...)
Affinity DataKi:  11.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM50087016(8-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5...)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM85749(III-BTD | NOCICEPTIN RECEPTOR ANTAGONIST PEPTIDE I...)
Affinity DataKi:  60.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM50087016(8-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5...)
Affinity DataKi:  148nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM50083230(1-((3R,4R)-1-Cyclooctylmethyl-3-hydroxymethyl-pipe...)
Affinity DataKi:  214nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM50083230(1-((3R,4R)-1-Cyclooctylmethyl-3-hydroxymethyl-pipe...)
Affinity DataKi:  229nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM50087016(8-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5...)
Affinity DataKi:  302nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM85748(H-PHE-(R)-GLY-GLY-PHE-THR-GLY-ALA-ARG-LYS-SER-ALA-...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM85748(H-PHE-(R)-GLY-GLY-PHE-THR-GLY-ALA-ARG-LYS-SER-ALA-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM85748(H-PHE-(R)-GLY-GLY-PHE-THR-GLY-ALA-ARG-LYS-SER-ALA-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Leicester Royal Infirmary

Curated by PDSP Ki Database
LigandPNGBDBM50083230(1-((3R,4R)-1-Cyclooctylmethyl-3-hydroxymethyl-pipe...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed