Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50037104
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108815(4-(2-Benzhydryloxy-ethyl)-1-(4-iodo-benzyl)-piperi...)
Affinity DataIC50:  0.960nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108818(4-(2-Benzhydryloxy-ethyl)-1-(4-vinyl-benzyl)-piper...)
Affinity DataIC50:  2.96nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108817(4-(2-Benzhydryloxy-ethyl)-1-(4-ethynyl-benzyl)-pip...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50098396(Benzhydryl-[2-(1-benzyl-piperidin-4-yl)-ethyl]-ami...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108823(4-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataIC50:  8.23nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataIC50:  10.6nMAssay Description:Inhibition of binding of 3[H] WIN-35 428 to Dopamine transporter (DAT) of rat striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108820(4-(2-Benzhydryloxy-ethyl)-1-(4-isopropenyl-benzyl)...)
Affinity DataIC50:  11.6nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108821(3-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataIC50:  14.3nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108824(4-(2-Benzhydryloxy-ethyl)-1-(3-methoxy-benzyl)-pip...)
Affinity DataIC50:  19.6nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108819(4-(2-Benzhydryloxy-ethyl)-1-(4-naphthalen-2-yl-ben...)
Affinity DataIC50:  26.9nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108816(3-(2-Benzhydryloxy-ethyl)-1-(4-isopropyl-benzyl)-p...)
Affinity DataIC50:  63.1nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108822(4-(2-Benzhydryloxy-ethyl)-1-(4-prop-1-ynyl-benzyl)...)
Affinity DataIC50:  65.1nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108825(4-(2-Benzhydryloxy-ethyl)-1-(4-naphthalen-1-yl-ben...)
Affinity DataIC50:  113nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataIC50:  132nMAssay Description:Inhibition of binding of [3H]- citalopram to Serotonin transporter (SERT) of rat cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108826(4-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataIC50:  240nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  266nMAssay Description:Inhibition of binding of 3[H] WIN-35 428 to Dopamine transporter (DAT) of rat striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108819(4-(2-Benzhydryloxy-ethyl)-1-(4-naphthalen-2-yl-ben...)
Affinity DataIC50:  393nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108824(4-(2-Benzhydryloxy-ethyl)-1-(3-methoxy-benzyl)-pip...)
Affinity DataIC50:  472nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)
Affinity DataIC50:  496nMAssay Description:Inhibition of binding of [3H]- nisoxatine to Norepinephrine transporter (NET) of rat cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108821(3-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataIC50:  678nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108818(4-(2-Benzhydryloxy-ethyl)-1-(4-vinyl-benzyl)-piper...)
Affinity DataIC50:  715nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  737nMAssay Description:Inhibition of binding of [3H]- citalopram to Serotonin transporter (SERT) of rat cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108817(4-(2-Benzhydryloxy-ethyl)-1-(4-ethynyl-benzyl)-pip...)
Affinity DataIC50:  760nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108820(4-(2-Benzhydryloxy-ethyl)-1-(4-isopropenyl-benzyl)...)
Affinity DataIC50:  832nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108819(4-(2-Benzhydryloxy-ethyl)-1-(4-naphthalen-2-yl-ben...)
Affinity DataIC50:  856nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108823(4-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataIC50:  924nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108821(3-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataIC50:  984nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108820(4-(2-Benzhydryloxy-ethyl)-1-(4-isopropenyl-benzyl)...)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108817(4-(2-Benzhydryloxy-ethyl)-1-(4-ethynyl-benzyl)-pip...)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108816(3-(2-Benzhydryloxy-ethyl)-1-(4-isopropyl-benzyl)-p...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108824(4-(2-Benzhydryloxy-ethyl)-1-(3-methoxy-benzyl)-pip...)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108815(4-(2-Benzhydryloxy-ethyl)-1-(4-iodo-benzyl)-piperi...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108822(4-(2-Benzhydryloxy-ethyl)-1-(4-prop-1-ynyl-benzyl)...)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108818(4-(2-Benzhydryloxy-ethyl)-1-(4-vinyl-benzyl)-piper...)
Affinity DataIC50:  1.47E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108825(4-(2-Benzhydryloxy-ethyl)-1-(4-naphthalen-1-yl-ben...)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108816(3-(2-Benzhydryloxy-ethyl)-1-(4-isopropyl-benzyl)-p...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50098396(Benzhydryl-[2-(1-benzyl-piperidin-4-yl)-ethyl]-ami...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108822(4-(2-Benzhydryloxy-ethyl)-1-(4-prop-1-ynyl-benzyl)...)
Affinity DataIC50:  2.41E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50098396(Benzhydryl-[2-(1-benzyl-piperidin-4-yl)-ethyl]-ami...)
Affinity DataIC50:  2.62E+3nMAssay Description:Concentration causing 50% Inhibition of binding of [3H]- nisoxatine to Norepinephrine transporter (NET).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108815(4-(2-Benzhydryloxy-ethyl)-1-(4-iodo-benzyl)-piperi...)
Affinity DataIC50:  2.92E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108826(4-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataIC50:  3.34E+3nMAssay Description:Inhibition of [3H]- nisoxatine binding to Norepinephrine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  3.53E+3nMAssay Description:Inhibition of binding of [3H]- nisoxatine to Norepinephrine transporter (NET) of rat cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108825(4-(2-Benzhydryloxy-ethyl)-1-(4-naphthalen-1-yl-ben...)
Affinity DataIC50:  4.16E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50108826(4-[4-(2-Benzhydryloxy-ethyl)-piperidin-1-ylmethyl]...)
Affinity DataIC50:  4.33E+3nMAssay Description:Inhibition of [3H]- citalopram binding to Serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed