Compile Data Set for Download or QSAR
maximum 50k data
Found 78 Enz. Inhib. hit(s) with all data for entry = 50011955
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112518(3-(3-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  0.0280nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112521(4-Amino-2-(3-{2-ethyl-6-[1-(1-imino-ethyl)-piperid...)
Affinity DataKi:  0.100nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112524(7-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy]...)
Affinity DataKi:  0.100nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112513(4-Amino-2-(3-{2-ethyl-5-[1-(1-imino-ethyl)-piperid...)
Affinity DataKi:  0.100nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112516(7-{5-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-2-isopr...)
Affinity DataKi:  0.200nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112494(7-{5-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-2-methy...)
Affinity DataKi:  0.300nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112514(3-(3-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  0.310nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112528(3-(3-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  0.400nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112526(3'-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  0.460nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112512(3-(3-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  1.30nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112529(4'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  2.20nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112516(7-{5-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-2-isopr...)
Affinity DataKi:  3nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112494(7-{5-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-2-methy...)
Affinity DataKi:  3nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50088957(7-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy]...)
Affinity DataKi:  4nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112524(7-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy]...)
Affinity DataKi:  5nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112523(7-{4-Dimethylamino-2-ethyl-5-[1-(1-imino-ethyl)-pi...)
Affinity DataKi:  5nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50088957(7-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy]...)
Affinity DataKi:  5nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112514(3-(3-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  6.90nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112530(7-{4-Amino-2-ethyl-5-[1-(1-imino-ethyl)-piperidin-...)
Affinity DataKi:  8nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112523(7-{4-Dimethylamino-2-ethyl-5-[1-(1-imino-ethyl)-pi...)
Affinity DataKi:  10nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112517(3-(3-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  13nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112519(({1-(7-Carbamimidoyl-naphthalen-2-ylmethyl)-2-ethy...)
Affinity DataKi:  15nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112510(4'-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  17nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112518(3-(3-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  21nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112508(4'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  22nMAssay Description:Tested in vitro for the selectivity against thrombin (IIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112530(7-{4-Amino-2-ethyl-5-[1-(1-imino-ethyl)-piperidin-...)
Affinity DataKi:  24nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112522(CHEMBL280769 | N-{1-(7-Carbamimidoyl-naphthalen-2-...)
Affinity DataKi:  25nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112528(3-(3-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  32nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112511(3'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  34nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112521(4-Amino-2-(3-{2-ethyl-6-[1-(1-imino-ethyl)-piperid...)
Affinity DataKi:  43nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112519(({1-(7-Carbamimidoyl-naphthalen-2-ylmethyl)-2-ethy...)
Affinity DataKi:  50nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112522(CHEMBL280769 | N-{1-(7-Carbamimidoyl-naphthalen-2-...)
Affinity DataKi:  50nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112527(3-(3-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  58nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112531(4-(3-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  64nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112526(3'-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  67nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112512(3-(3-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  73nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112529(4'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  73nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112525(4-(3-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  74nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112521(4-Amino-2-(3-{2-ethyl-6-[1-(1-imino-ethyl)-piperid...)
Affinity DataKi:  75nMAssay Description:Tested in vitro for the selectivity against thrombin (IIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112508(4'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  91nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112513(4-Amino-2-(3-{2-ethyl-5-[1-(1-imino-ethyl)-piperid...)
Affinity DataKi:  120nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112517(3-(3-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  130nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112510(4'-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  140nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112515(4'-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  150nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112509(3'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  150nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112508(4'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  180nMAssay Description:Tested in vitro for the inhibitory potency against Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112511(3'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  190nMAssay Description:Tested in vitro for the selectivity against thrombin (IIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112511(3'-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  190nMAssay Description:Tested in vitro for the selectivity against trypsin (Trp)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112518(3-(3-{2-Ethyl-6-[1-(1-imino-ethyl)-piperidin-4-ylo...)
Affinity DataKi:  200nMAssay Description:Tested in vitro for the selectivity against thrombin (IIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50112510(4'-{2-Ethyl-5-[1-(1-imino-ethyl)-piperidin-4-yloxy...)
Affinity DataKi:  210nMAssay Description:Tested in vitro for the selectivity against thrombin (IIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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