Compile Data Set for Download or QSAR
maximum 50k data
Found 47 Enz. Inhib. hit(s) with all data for entry = 50013184
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127518(CHEMBL57104 | peptidomimetic)
Affinity DataEC50:  0.190nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127553(2-(2-1H-Indol-2-yl-acetylamino)-pentanedioic acid ...)
Affinity DataEC50:  57nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127520(CHEMBL57438 | peptidomimetic)
Affinity DataEC50:  1.5nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127519(CHEMBL262992 | [D-Tyr6-, Beta-Ala11, Phe13, Nle14]...)
Affinity DataEC50:  310nMAssay Description:Effective concentration required against nueromedin B receptor (NMB-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127522(2-Phenylacetylamino-pentanedioic acid 5-amide 1-{[...)
Affinity DataEC50:  1.91E+4nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127521(CHEMBL57046 | peptidomimetic)
Affinity DataEC50:  2.70E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127525(2-Benzylamino-N-[2-(1H-indol-3-yl)-1-phenethylcarb...)
Affinity DataEC50:  46nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127523(3-(1H-Indol-3-yl)-N-phenethyl-2-{2-[(pyridin-3-ylm...)
Affinity DataEC50:  21nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127524(CHEMBL58097 | peptidomimetic)
Affinity DataEC50:  7.90E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127526(CHEMBL56562 | peptidomimetic)
Affinity DataEC50:  15nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127527(CHEMBL294647 | peptidomimetic)
Affinity DataEC50:  2.20nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127528(3-(1H-Indol-3-yl)-N-phenethyl-2-[2-(2-1,2,3,4-tetr...)
Affinity DataEC50:  310nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127519(CHEMBL262992 | [D-Tyr6-, Beta-Ala11, Phe13, Nle14]...)
Affinity DataEC50:  84nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127529(2-[2-(4-Chloro-benzylamino)-acetylamino]-3-(1H-ind...)
Affinity DataEC50:  2.90nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127530(2-[2-(2-Benzo[1,3]dioxol-5-yl-acetylamino)-propion...)
Affinity DataEC50:  7.80nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127531(CHEMBL292227 | N-[2-(1H-Indol-3-yl)-1-phenethylcar...)
Affinity DataEC50:  25nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127532(CHEMBL438926 | Val-Pro-Leu-Pro-Ala-Gly-Gly-Gly-Thr...)
Affinity DataEC50:  3.20E+3nMAssay Description:Effective concentration required against nueromedin B receptor (NMB-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127532(CHEMBL438926 | Val-Pro-Leu-Pro-Ala-Gly-Gly-Gly-Thr...)
Affinity DataEC50:  6.40E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127534(CHEMBL56626 | peptidomimetic)
Affinity DataEC50:  6nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127533(2-(2-Amino-3-phenyl-propionylamino)-pentanedioic a...)
Affinity DataEC50:  710nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127522(2-Phenylacetylamino-pentanedioic acid 5-amide 1-{[...)
Affinity DataEC50:  1.50E+4nMAssay Description:Effective concentration required against nueromedin B receptor (NMB-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127522(2-Phenylacetylamino-pentanedioic acid 5-amide 1-{[...)
Affinity DataEC50:  1.20E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127535(2-[2-(4-Chloro-phenyl)-acetylamino]-pentanedioic a...)
Affinity DataEC50:  1.40E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127536(2-[2-(4-Benzyl-piperidin-1-yl)-acetylamino]-3-(1H-...)
Affinity DataEC50:  30nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127538(CHEMBL291549 | peptidomimetic)
Affinity DataEC50:  240nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127540(CHEMBL175651 | peptidomimetic)
Affinity DataEC50:  19nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127537(3-(1H-Indol-3-yl)-2-[2-(2-1H-indol-2-yl-acetylamin...)
Affinity DataEC50:  79nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127539(3-(1H-Indol-3-yl)-N-phenethyl-2-(2-phenylacetylami...)
Affinity DataEC50:  2.10nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50071745(CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Trp-Ala-...)
Affinity DataEC50:  41nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127541(CHEMBL418147 | peptidomimetic)
Affinity DataEC50:  24nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127542(2-{2-[2-(4-Chloro-phenyl)-acetylamino]-propionylam...)
Affinity DataEC50:  140nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127535(2-[2-(4-Chloro-phenyl)-acetylamino]-pentanedioic a...)
Affinity DataEC50:  1.22E+4nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127543(3-(1H-Indol-3-yl)-N-phenethyl-2-[2-(2-pyridin-3-yl...)
Affinity DataEC50:  32nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127544(CHEMBL56369 | peptidomimetic)
Affinity DataEC50:  1.40nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127545(2-[3-(4-Chloro-phenyl)-propionylamino]-pentanedioi...)
Affinity DataEC50:  230nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127546(2-{2-[3-(4-Chloro-phenyl)-propionylamino]-propiony...)
Affinity DataEC50:  6.40E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127548(2-(2-Benzylamino-acetylamino)-3-(1H-indol-3-yl)-N-...)
Affinity DataEC50:  21nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127535(2-[2-(4-Chloro-phenyl)-acetylamino]-pentanedioic a...)
Affinity DataEC50:  1.85E+4nMAssay Description:Effective concentration required against nueromedin B receptor (NMB-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127532(CHEMBL438926 | Val-Pro-Leu-Pro-Ala-Gly-Gly-Gly-Thr...)
Affinity DataEC50:  34nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50071745(CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Trp-Ala-...)
Affinity DataEC50:  4.50E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127547(CHEMBL57559 | peptidomimetic)
Affinity DataEC50:  3.10nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127551(CHEMBL292646 | peptidomimetic)
Affinity DataEC50:  9.30nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50071745(CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Trp-Ala-...)
Affinity DataEC50:  120nMAssay Description:Effective concentration required against nueromedin B receptor (NMB-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127550(3-(1H-Indol-3-yl)-N-phenethyl-2-(2-phenethylamino-...)
Affinity DataEC50:  17nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127552(2-[2-(4-Benzyl-piperazin-1-yl)-acetylamino]-3-(1H-...)
Affinity DataEC50:  70nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127549(2-(4-Chloro-benzylamino)-N-[2-(1H-indol-3-yl)-1-ph...)
Affinity DataEC50:  4nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127519(CHEMBL262992 | [D-Tyr6-, Beta-Ala11, Phe13, Nle14]...)
Affinity DataEC50:  151nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed