Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50000176
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002461(10-Ethyl-1-[2-(3-ethyl-3H-benzothiazol-2-ylidene)-...)
Affinity DataIC50:  180nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002464(10-Ethyl-1-[2-(1,1,3-trimethyl-1,3-dihydro-benzo[e...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002460(1,3-Diethyl-2-[3-(3-ethyl-3H-benzooxazol-2-ylidene...)
Affinity DataIC50:  310nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002456(1,3-Diethyl-2-[3-(3-ethyl-3H-benzothiazol-2-yliden...)
Affinity DataIC50:  320nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002459(1,3-Diethyl-2-[3-(1-ethyl-3,3-dimethyl-1,3-dihydro...)
Affinity DataIC50:  360nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002458(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataIC50:  390nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002457(1-(2-Acetoxy-ethyl)-3-ethyl-2-[3-(1,3,3-trimethyl-...)
Affinity DataIC50:  410nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002452(3-Ethyl-1-(2-hydroxy-ethyl)-2-[3-(1,3,3-trimethyl-...)
Affinity DataIC50:  450nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002454(CHEMBL386306 | D-Lys(Nicotinoyl)-Pro(3-Pyridyl)-Al...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataIC50:  510nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002455(10-Ethyl-1-[2-(1,3,3-trimethyl-1,3-dihydro-indol-2...)
Affinity DataIC50:  790nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002451(5-Ethyl-4-[2-(3-ethyl-3H-benzothiazol-2-ylidene)-e...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002463(1,3-Diethyl-2-[3-(1-methyl-1H-benzo[cd]indol-2-yli...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Rochester

Curated by ChEMBL
LigandPNGBDBM50002453(10-Ethyl-1-[2-(3-ethyl-3H-benzooxazol-2-ylidene)-e...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of Tachykinin receptor 1 of rat forebrain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed