Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50041996
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50366785(NELFINAVIR)
Affinity DataIC50:  1.25E+4nMAssay Description:TP_TRANSPORTER: increase in mitoxantrone intracellular accumulation in BCRP-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM519((2S)-N-[(2S,3R)-4-[(3S,4aS,8aS)-3-(tert-butylcarba...)
Affinity DataIC50:  1.95E+4nMAssay Description:TP_TRANSPORTER: increase in mitoxantrone intracellular accumulation in BCRP-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
University Of Washington

Curated by ChEMBL
LigandPNGBDBM520(1,3-thiazol-5-ylmethyl N-[(2S,3S,5S)-3-hydroxy-5-[...)
Affinity DataIC50:  1.95E+4nMAssay Description:TP_TRANSPORTER: increase in mitoxantrone intracellular accumulation in BCRP-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed