Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50037307
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122294(CHEMBL292092 | N-(5-fluoro-2-phenoxyphenyl)-N-(2-(...)
Affinity DataKi:  0.0780nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.160nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122295(CHEMBL63065 | N-(2-Fluoromethoxy-5-methoxy-benzyl)...)
Affinity DataKi:  0.170nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  0.830nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50144889(CHEMBL72521 | N-(5-Fluoro-2-phenoxy-phenyl)-N-(2-i...)
Affinity DataKi:  4.80nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50144887(CHEMBL443526 | Toluene-4-sulfonic acid 2-(2-{[acet...)
Affinity DataKi:  18.1nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed