Affinity DataKi: 0.600nMAssay Description:Binding affinity for adenosine A2a receptor by using as [3H]-ZM-241,385 radioligand in membranes from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX iradioligand n membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against Adenosine A2b receptor labeled by [3H]-ZM-241,385 in membranes prepared from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity against Adenosine A3 receptor by displacement of specific binding of [125I]-AB-MECA in membranes prepared from CHO-A3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity against Adenosine A1 receptor labeled by [3H]-CPX in membranes prepared from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity for adenosine A3 receptor by displacement of specific binding of [125I]-AB-MECA in membranes from CHO-A3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >23nMAssay Description:Binding affinity for adenosine A2a receptor labeled by [3H]-ZM-241,385 in membranes from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity against Adenosine A2a receptor labeled by [3H]-ZM-241,385 in membranes prepared from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity for adenosine A3 receptor by displacement of specific binding of [125I]-AB-MECA in membranes from CHO-A3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 127nMAssay Description:Binding affinity against Adenosine A2b receptor labeled by [3H]-ZM-241,385 in membranes prepared from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 127nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: >167nMAssay Description:Binding affinity against Adenosine A3 receptor by displacement of specific binding of [125I]-AB-MECA in membranes prepared from CHO-A3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >200nMAssay Description:Binding affinity against Adenosine A1 receptor labeled by [3H]-CPX in membranes prepared from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: >200nMAssay Description:Binding affinity against Adenosine A2a receptor labeled by [3H]-ZM-241,385 in membranes prepared from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 207nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Binding affinity against Adenosine A1 receptor labeled by [3H]-CPX in membranes prepared from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 215nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 215nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 255nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: >260nMAssay Description:Binding affinity against Adenosine A2a receptor labeled by [3H]-ZM-241,385 in membranes prepared from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 288nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: >290nMAssay Description:Binding affinity against Adenosine A3 receptor by displacement of specific binding of [125I]-AB-MECA in membranes prepared from CHO-A3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 325nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Binding affinity for adenosine A2a receptor by using as [3H]-ZM-241,385 (2 nM) radioligand in membranes from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 438nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 473nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 485nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 526nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 557nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 643nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 645nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 945nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Binding affinity for adenosine A2a receptor by using as [3H]-ZM-241,385 (2 nM) radioligand in membranes from HEK-A2A cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.12E+3nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.16E+3nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+3nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.68E+3nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.83E+3nMAssay Description:Binding affinity for adenosine A1 receptor by using as [3H]-CPX (0.5 nM) radioligand in membranes from Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.83E+3nMAssay Description:Binding affinity for adenosine A2b receptor by using as [3H]-ZM-241,385 (14 nM) radioligand in membranes from HEK-A2B cellsMore data for this Ligand-Target Pair