Compile Data Set for Download or QSAR
maximum 50k data
Found 82 Enz. Inhib. hit(s) with all data for entry = 50017228
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataIC50:  92nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179235(2-{5-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  105nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179229(2-{5-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataIC50:  120nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179225(2-{4-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataIC50:  127nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179236(2-(5-(3-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataIC50:  152nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179227(2-(5-(2-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataIC50:  422nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179240(3-{5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  584nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179226(2-{5-[3-(3-cyano-7-propyl-1H-indol-6-yloxy)propoxy...)
Affinity DataIC50:  759nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179233(2-{4-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  774nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179234(2-{6-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  1.05E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179243(2-{5-[5-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  1.05E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179248(3-{4-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179231(CHEMBL198929 | {5-[3-(7-propyl-3-trifluoromethylbe...)
Affinity DataIC50:  1.12E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179249(2-ethyl-2-{4-[3-(7-propyl-3-trifluoromethylbenzo[d...)
Affinity DataIC50:  1.28E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179238(2-{4-[2-methyl-3-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179244(2-{5-[3-methyl-5-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataIC50:  1.37E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179239(2-{4-[3-methyl-5-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataIC50:  1.45E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179241(2-{4-[2-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179246(2-{4-[3-(2-phenyl-7-propyl-1H-indol-6-yloxy)propox...)
Affinity DataIC50:  1.68E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179230(2-ethyl-2-{5-[3-(7-propyl-3-trifluoromethylbenzo[d...)
Affinity DataIC50:  1.71E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179247(2-{4-[5-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  1.78E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179232(2-{4-[3-(2-phenyl-7-propylbenzo[b]furan-6-yloxy)pr...)
Affinity DataIC50:  1.95E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179237(2-{4-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50:  1.99E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179245(2-(5-{3-[3-(2,2,2-trifluoroethyl-1-one)-7-propyl-1...)
Affinity DataIC50:  2.41E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179242(2-{4-[3-(3-phenyl-7-propylbenzo[b]furan-6-yloxy)pr...)
Affinity DataIC50:  3.97E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179228(2-{5-[3-(7-propyl-1H-indol-6-yl)propoxy]indol-1-yl...)
Affinity DataIC50:  4.81E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179225(2-{4-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataEC50:  2nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179226(2-{5-[3-(3-cyano-7-propyl-1H-indol-6-yloxy)propoxy...)
Affinity DataEC50:  5.21E+3nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179227(2-(5-(2-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataEC50:  690nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179228(2-{5-[3-(7-propyl-1H-indol-6-yl)propoxy]indol-1-yl...)
Affinity DataEC50:  1.81E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179230(2-ethyl-2-{5-[3-(7-propyl-3-trifluoromethylbenzo[d...)
Affinity DataEC50:  5.90E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179232(2-{4-[3-(2-phenyl-7-propylbenzo[b]furan-6-yloxy)pr...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179233(2-{4-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179236(2-(5-(3-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataEC50:  14nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179228(2-{5-[3-(7-propyl-1H-indol-6-yl)propoxy]indol-1-yl...)
Affinity DataEC50:  420nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179229(2-{5-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataEC50:  80nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179237(2-{4-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  610nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179238(2-{4-[2-methyl-3-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataEC50:  3.03E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179235(2-{5-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  243nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179237(2-{4-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  186nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179239(2-{4-[3-methyl-5-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179240(3-{5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  1.20E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179233(2-{4-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179243(2-{5-[5-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  1.49E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179242(2-{4-[3-(3-phenyl-7-propylbenzo[b]furan-6-yloxy)pr...)
Affinity DataEC50:  169nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  220nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179245(2-(5-{3-[3-(2,2,2-trifluoroethyl-1-one)-7-propyl-1...)
Affinity DataEC50:  9.17E+3nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179234(2-{6-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  1.82E+3nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179232(2-{4-[3-(2-phenyl-7-propylbenzo[b]furan-6-yloxy)pr...)
Affinity DataEC50:  7.74E+3nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179234(2-{6-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  80nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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