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Found 29 Enz. Inhib. hit(s) with all data for entry = 50017648
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  70nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185034(CHEMBL382444 | N-arachidonoyl-O-(2-hydroxyethyl)hy...)
Affinity DataKi:  81nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  180nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185034(CHEMBL382444 | N-arachidonoyl-O-(2-hydroxyethyl)hy...)
Affinity DataKi:  470nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM29080(CHEMBL280065 | N-oleoylethanolamine | Oleamide MEA...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185035(CHEMBL204403 | N-arachidonoyl-N-(2-hydroxyethyl)hy...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185037(CHEMBL203380 | O-arachidonoyl-N-(2-hydroxyethyl)hy...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185037(CHEMBL203380 | O-arachidonoyl-N-(2-hydroxyethyl)hy...)
Affinity DataKi:  3.50E+3nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185033(CHEMBL208270 | N-oleoyl-O-(2-hydroxyethyl)hydroxyl...)
Affinity DataKi:  3.80E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185035(CHEMBL204403 | N-arachidonoyl-N-(2-hydroxyethyl)hy...)
Affinity DataKi:  3.90E+3nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185031(CHEMBL203189 | N-oleoyl-N-(2-hydroxyethyl)hydroxyl...)
Affinity DataKi:  5.40E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185030(CHEMBL380925 | O-oleoyl-N-(2-hydroxyethyl)hydroxyl...)
Affinity DataKi:  8.60E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185036(CHEMBL205609 | N-palmitoyl-O-(2-hydroxyethyl)hydro...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185036(CHEMBL205609 | N-palmitoyl-O-(2-hydroxyethyl)hydro...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM29080(CHEMBL280065 | N-oleoylethanolamine | Oleamide MEA...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185031(CHEMBL203189 | N-oleoyl-N-(2-hydroxyethyl)hydroxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185030(CHEMBL380925 | O-oleoyl-N-(2-hydroxyethyl)hydroxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185029(CHEMBL205272 | O-palmitoyl-N-(2-hydroxyethyl)hydro...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185033(CHEMBL208270 | N-oleoyl-O-(2-hydroxyethyl)hydroxyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185032(CHEMBL206425 | N-palmitoyl-N-(2-hydroxyethyl)hydro...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185032(CHEMBL206425 | N-palmitoyl-N-(2-hydroxyethyl)hydro...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185029(CHEMBL205272 | O-palmitoyl-N-(2-hydroxyethyl)hydro...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185032(CHEMBL206425 | N-palmitoyl-N-(2-hydroxyethyl)hydro...)
Affinity DataEC50:  600nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM29080(CHEMBL280065 | N-oleoylethanolamine | Oleamide MEA...)
Affinity DataEC50:  890nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185031(CHEMBL203189 | N-oleoyl-N-(2-hydroxyethyl)hydroxyl...)
Affinity DataEC50:  400nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185034(CHEMBL382444 | N-arachidonoyl-O-(2-hydroxyethyl)hy...)
Affinity DataEC50:  250nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185033(CHEMBL208270 | N-oleoyl-O-(2-hydroxyethyl)hydroxyl...)
Affinity DataEC50:  320nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185035(CHEMBL204403 | N-arachidonoyl-N-(2-hydroxyethyl)hy...)
Affinity DataEC50:  260nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataEC50:  490nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed