Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50000572
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  1.60nMAssay Description:Opioid receptor activity in terms of inhibition of [3H]-dihydromorphine binding in rat brain membraneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50:  4.20nMAssay Description:Neuroleptic activity in terms of [3H]-spiroperidol binding in rat striatal membraneto Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50007421(CHEMBL59245 | Propionic acid 1-[4-(4-fluoro-phenyl...)
Affinity DataIC50:  6.10nMAssay Description:Opioid activity in terms of inhibition of [3H]-dihydromorphine binding to opioid receptor mu in rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50007421(CHEMBL59245 | Propionic acid 1-[4-(4-fluoro-phenyl...)
Affinity DataIC50:  9.5nMAssay Description:Opioid activity in terms of inhibition of [3H]-dihydromorphine binding to Opioid receptor mu 1 in rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50007421(CHEMBL59245 | Propionic acid 1-[4-(4-fluoro-phenyl...)
Affinity DataIC50:  43nMAssay Description:Neuroleptic activity in terms of [3H]-spiroperidol binding to dopamine receptor D2 in rat striatal membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50007421(CHEMBL59245 | Propionic acid 1-[4-(4-fluoro-phenyl...)
Affinity DataIC50:  54nMAssay Description:Neuroleptic activity in terms of [3H]-spiroperidol binding to Dopamine receptor D2 in rat striatal membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50007420(CHEMBL418289 | Propionic acid 1-[4-(4-fluoro-pheny...)
Affinity DataIC50:  147nMAssay Description:Neuroleptic activity in terms of [3H]-spiroperidol binding to Dopamine receptor D2 in rat striatal membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataIC50:  302nMAssay Description:Neuroleptic activity in terms of [3H]-spiroperidol binding in rat striatal membrane to Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM50007420(CHEMBL418289 | Propionic acid 1-[4-(4-fluoro-pheny...)
Affinity DataIC50:  1.79E+3nMAssay Description:Opioid activity in terms of inhibition of [3H]-dihydromorphine binding to Opioid receptor mu 1 in rat brain membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Istituto Superiore Di Sanità

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataIC50:  3.05E+3nMAssay Description:Neuroleptic activity in terms of [3H]-spiroperidol binding in rat striatal membrane to Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed